Publications

162. Wilson, R. M.; Thalji, R. K.; Bergman, R. G.; Ellman, J. A.
Enantioselective Synthesis of a PKC Inhibitor via Catalytic C-H Bond Activation
Org. Lett.  2006, 8, 1745-1747.
161. Beenen, M. A.; Weix, D. J.; Ellman, J. A.
Asymmetric Synthesis of Protected Arylglycines by Rhodium-Catalyzed Addition of Arylboronic Acids to N-tert-Butanesulfinyl Imino Esters
J. Am. Chem. Soc.  2006, 128, 6304-6305.
Write-up in Organic Process Research and Development
160. Colby, D. A.; Bergman, R. G.; Ellman, J. A.
Stereoselective Alkylation of alpha,beta-Unsaturated Imines via C-H Bond Activation
J. Am. Chem. Soc.  2006, 128,  5604-05.
159. Lewis, J. C.; Wu, J. Y.; Ellman, J. A.; Bergman, R. G.
Microwave-Promoted Rhodium-Catalyzed Arylation of Heterocycles through CH Bond Activation
Angew. Chem. Int. Ed.  2006, 45, 1589-1591.
158. Wiedemann, S. H.; Lewis, J. C.; Ellman, J. A.; Bergman, R. G.
Experimental and Computational Studies on the Mechanism of N-Heterocycle C-H Activation by Rh(I)
J. Am. Chem. Soc.   2006, 128, 2452-2462.
157. Wiedemann, S. H.; Ellman, J. A.; Bergman, R. G.
Rhodium-Catalyzed Direct C-H Addition of 3,4-Dihydroquinazolines to Alkenes and Their Use in the Total Synthesis of Vasicoline
J. Org. Chem.  2006, 71, 1969-1976.
Write-up in Organic Process Research and Development
156. Wood, W. J. L.; Patterson, A. W.; Tsuruoka, H.; Jain, R. K.; Ellman, J. A
Substrate Activity Screening: A Fragment-Based Method for the Rapid Identification of Nonpeptidic Protease Inhibitors
J. Am. Chem. Soc.  2005, 127, 5521-15527.
Research Highlight in Nature Chemical Biology
155. McMahon, J. P.; Ellman, J. A.
Asymmetric Conjugate Addition of Copper Reagents to alpha,beta-Unsaturated tert-Butanesulfinyl Imines
Org. Lett.  2005, 7, 5393-5396.
154. Weix, D. J.; Ellman, J. A.
(+)-2-Methyl-2-propanesulfinamide
Org. Synth.  2005, 82, 157-165.
153. Lewis, J. C.; Wu, J.; Bergman, R. G.; Ellman, J. A.
Preagostic Rh-H Interactions and C-H Bond Functionalization: A Combined Experimental and Theoretical Investigation of Rhodium(I) Phosphinite Complexes
Organometallics  2005, 24, 5737-5746.
152. O'Malley, S. J.; Tan, K. L.; Watzke, A.; Bergman, R. G.; Ellman, J. A.
Total Synthesis of (+)-Lithospermic Acid by Asymmetric Intramolecular Alkylation via Catalytic C-H Bond Activation
J. Am. Chem. Soc  2005, 127, 13496-13497.
151. Peltier, H. M.; Ellman, J. A.
N-Sulfinyl Metalloenamine Conjugate Additions: Asymmetric Synthesis of Piperidines
J. Org. Chem.  2005, 70, 7342-7345.
150. Thalji, R. K.; Ahrendt, K. A.; Bergman, R. G.; Ellman, J. A.
Annulation of Aromatic Imines via Directed C-H Bond Activation
J. Org. Chem.  2005, 70, 6775-6781.
149. Brinner, K. M.; Ellman, J. A.
A Rapid and General Method for the Asymmetric Synthesis of 2-Substituted Pyrrolidines Using tert-Butanesulfinamide
Org. Biomol. Chem.  2005, 3, 2109-2113.
148. Ghosalia, D. N.; Salisbury, C. M.; Maly, D. J.; Ellman, J. A.; Diamond, S. L.
Profiling Serine Protease Substrate Specificity with Solution Phase Fluorogenic Peptide Microarrays
Proteomics  2005, 5, 1292-1298.
147. Wiedemann, S. H.; Ellman, J. A.; Bergman, R. G.
Catalytic Functionalization of N-Heterocycles via their Rhodium-Carbene Complexes.
In Handbook of C-H Transformations; Dyker, G., Ed.: Wiley-VCH Verlag GmbH & Co. KGaA; Weinheim,  2005, , 187-193.
146. Gosalia, D. N.; Salisbury, C. M.; Ellman, J. A.; Diamond, S. L.
High Throughput Substrate Specificity Profiling of Serine and Cysteine Proteases Using Solution-Phase Fluorogenic Peptide Microarays
Molec. Cell. Proteomics  2005, 4, 626-636.
145. Peltier, H. M.; Evans, J. W.; Ellman, J. A.
Catalytic Enantioselective Sulfinyl Transfer Using Cinchona Alkaloid Catalysts
Org. Lett.  2005, 7, 1733-1736.
144. Brinner, K.; Ellman, J. A.
“Asymmetric Synthesis of  ß-Amino Acids by Enolate Additions to tert-Butanesulfinyl Imines” In Enantioselective  Synthesis of ß-Amino Acids, 2nd Edition; Juaristi, E., Soloshonok, V.,  Eds.; John Wiley & Sons, Hoboken, NJ;
  2005, , 181-194.
143. Brinner, K. M.; Powles, M. A.; Schmatz, D. M.; Ellman, J. A.
Potent 4-Aminopiperidine Based Antimalarial Agents
Bioorg. Med. Chem. Lett.  2005, 15, 345-348.
142. Weix, D. J.; Shi, Y.; Ellman, J. A.
Diastereoselective and Enantioselective Rh(I)-Catalyzed Additions of Arylboronic Acids to N-tert-Butanesulfinyl and N-Diphenylphosphinoyl Aldimines
J. Am. Chem. Soc.  2005, 127, 1092-1093.
141. Kochi , T.; Ellman, J. A.
Asymmetric alpha-Alkylation of N’-tert-Butanesulfinyl Amidines. Application to the Total Synthesis of (6R,7S)-7-Amino-7,8-dihydro-alpha-bisabolene
J. Am. Chem. Soc.  2004, 126, 15652-15653.
140. Tan, K. L.; Park, S.; Ellman, J. A.; Bergman, R. G.
Intermolecular Coupling of Alkenes to Heterocycles via C-H Bond Activation
J. Org. Chem.  2004, 69, 7329-7335.
139. Evans, J .W.; Fierman, M. B.; Miller, S. J.; Ellman, J. A.
Catalytic Enantioselective Synthesis of Sulfinate Esters Through the Dynamic Resolution of tert-Butanesulfinyl Chloride
J. Am. Chem. Soc.  2004, 126, 8134-8135.
138. Schenkel, L. B.; Ellman, J. A.
Self-Condensation of N-tert-Butanesulfinyl Aldimines: Application to the Asymmetric Synthesis of Biologically Important Amine-Containing Compounds
Org. Lett.  2004, 6, 3621-3624.
137. Klei, S. R.; Tan, K. L.; Golden, J. T.; Yung, C. M.; Thalji, R. K.; Ahrendt, K. A.; Ellman, J. A.; Tilley, T. D.; Bergman, R. G.
C-H Bond activation by iridium and rhodium complexes: Catalytic hydrogen-deuterium exchange and C-C bond-forming reactions. In Activation and Functionalization of C-H Bonds; Goldberg, K. I.; Goldman, A. S., Ed.; ACS Symposium Series 885; American Chemical Society; Washington, DC,
  2004, , 46-55.
136. Thalji, R. K.; Ellman, J. A.; Bergman, R. G.
Highly Efficient and Enantioselective Cyclization of Aromatic Imines via Directed C-H Bond Activation
J. Am. Chem. Soc.  2004, 126, 7192-7193.
135. Kochi , T.; Mukade, T.
Asymmetric Synthesis of Amines with tert-Butanesulfinamide and Its Application
J. Syn. Org. Chem. Jpn.  2004, 62, 128-139.
134. McMahon, J. P.; Ellman, J. A.
Highly Stereoselective Addition of Organometallic Reagents to N-tert-Butanesulfinyl Imines Derived from 3- and 4-Substituted Cyclohexanones
Org. Lett.  2004, 6, 1645-1647.
133. Wiedemann, S. H.; Bergman, R. G.; Ellman, J. A.
Rhodium-Catalyzed Direct C-H Addition of 4,4-Dimethyl-2-oxazoline to Alkenes
Org. Lett.  2004, 6, 1685-1687.

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