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209. |
Drag, M.; Bogyo, M.; Ellman, J. A.; Salvesen, G. S.
Aminopeptidase Fingerprints, an Integrated Approach for Identification of Good Substrates and Optimal Inhibitors
J. Biol. Chem. 2010, 285, 3310-3318.
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208. |
Sun, C.; Su, K.-H.; Valentine, J.; Rosa-Bauza, Y. T.; Ellman, J. A.; Elboudwarej, O.; Mukherjee, B.; Craik, C. S.; Shuman, M. A.; Chen, F. F.; Zhang, X.
Time-Resolved Single-Step Protease Activity Quantification Using Nanoplasmonic Resonator Sensors
ACS Nano 2010, 4, 978–984.
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207. |
Colby, D. A.; Bergman, R. G.; Ellman, J. A.
Rhodium-Catalyzed C-C Bond Formation via Heteroatom-Directed C-H Bond Activation
Chem. Rev. 2010, 110, 624-655.
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206. |
Storgaard, M.; Ellman, J. A.
Rhodium-Catalyzed Enantioselective Addition of Arylboronic Acids to In Situ Generated N-Boc Arylimines. Preparation of (S)-tert-Butyl (4-Chlorophenyl)(Thiophen-2-yl-MethyylCarbamate
Org. Synth. 2009, 86, 360-373.
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205. |
Rawls, K. A.; Lang, T. P.; Takeuchi, J.; Imamura, S.; Baguley, T. D.; Grundner, C.; Alber, T.; Ellman, J. A.
Fragment-based discovery of selective inhibitors of the Mycobacterium tuberculosis protein tyrosine phosphatase PtpA
Bioorg. Med. Chem. Lett. 2009, 19, 6851-6854.
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204. |
Kimmel, K. L.; Robak, M. T.; Ellman, J. A.
Enantioselective Addition of Thioacetic Acid to Nitroalkenes via N-Sulfinyl Urea Organocatalysis
J. Am. Chem. Soc. 2009, 131, 8754–8755.
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203. |
Arceo, E.; Marsden, P.; Bergman, R. G.; Ellman, J. A.
An Efficient Didehydroxylation Method for the Biomass-Derived Polyols Glycerol and Erythritol. Mechanistic Studies of a Formic Acid-Mediated Deoxygenation
Chem. Commun. 2009, , 3357-3359.
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202. |
Tsai, A. S.; Wilson, R. M.; Hirada, H.; Bergman, R. G.; Ellman, J. A.
Rhodium Catalyzed Enantioselective Cylization of Substituted Imidazoles via C–H Bond Activation
Chem. Commun. 2009, , 3910-3912.
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201. |
Brak, K.; Harris, K. ; Ellman, J. A.
General One-pot Method for the Preparation of N-tert-Butanesulfinyl Amine Diastereomer Mixtures as Standards for Stereoselectivity Determinations
J. Org. Chem. 2009, 74, 3606-3608.
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200. |
Brak, K.; Ellman, J. A.
Asymmetric Synthesis of α–Branched Allylic Amines by the Rh(I)-Catalyzed Addition of Alkenyltrifluoroborates to N-tert-Butanesulfinyl Aldimines
J. Am. Chem. Soc. 2009, 131, 3850–3851.
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199. |
Yotphan, S.; Bergman, R. G.; Ellman, J. A.
Application of Daugulis Copper-Catalyzed Direct Arylation to the Synthesis of 5-Aryl Benzotriazepines
Org. Lett. 2009, 11, 1511–1514.
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198. |
Wakayama , M.; Ellman, J. A.
Recycling the tert-Butanesulfinyl Group in the Synthesis of Amines Using tert-ButanesulfinamideRecycling the tert-Butanesulfinyl Group in the Synthesis of Amines Using tert-Butanesulfinamide
J. Org. Chem. 2009, 74, 2646–2650.
Write-up in Organic Process Research and Development
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197. |
Berman, A. M.; Lewis, J. C.; Bergman, R. G.; Ellman, J. A.
Rh(I)-Catalyzed Direct Arylation of Pyridines and Quinolines
J. Am. Chem. Soc. 2008, 130, 14926–14927.
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196. |
Harada, H.; Thalji, R. K.; Bergman, R. G.; Ellman, J. A.
Enantioselective Intramolecular Hydroarylation of Alkenes via Directed C-H Bond Activation
J. Org. Chem. 2008, 73, 6772-6779.
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195. |
Lewis, J. C.; Bergman, R. G.; Ellman, J. A.
Direct Functionalization of Nitrogen Heterocycles via Rh-Catalyzed C-H Bond Activation
Acc. Chem. Res. 2008, 41, 1013-1025.
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194. |
Drag, M.; Mikolajczyk, J.; Bekes, M.; Reyes-Turcu, F.; Ellman, J. A.; Wilkinson, K. D.; Salvesen, G. S.
Positional-Scanning Fluorogenic Substrate Libraries Reveal Unexpected Specificity Determinants of Deubiquitinating Enzymes (DUBs)
Biochem. J. 2008, 415, 367-375.
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193. |
Trincado, M.; Ellman, J. A.
Enantioselective Synthesis of alpha-Aryl Alkylamines by Rh-Catalyzed Addition Reactions of Arylboronic Acids to Aliphatic Imines
Angew. Chem. Int. Ed. 2008, 47, 5623-5626.
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192. |
Beenen, M. A.; An, C.; Ellman, J. A.
Asymmetric Copper-Catalyzed Synthesis of alpha-Amino Boronate Esters from N-tert-Butanesulfinyl Aldimines
J. Am. Chem. Soc. 2008, 130, 6910-6911.
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191. |
Patterson, A. W.; Peltier, H. M.; Ellman, J. A.
Expedient Synthesis of N-Methyl Tubulysin Analogues with High Cytotoxicity
J. Org. Chem. 2008, 73, 4362-4369.
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190. |
Gribble, M. W.; Ellman, J. A.; Bergman, R. G.
Synthesis of a Benzodiazepine-Derived Rhodium NHC Complex by C-H Bond Activation
Organometallics 2008, 27, 2152-2155.
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189. |
Brak, K.; Doyle, P. S.; McKerrow, J. H.; Ellman, J. A.
Identification of a New Class of Nonpeptidic Inhibitors of Cruzain
J. Am. Chem. Soc. 2008, 130, 6404-6410.
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188. |
Tsai, A. S.; Bergman, R. G.; Ellman, J. A.
Asymmetric Synthesis of (−)-Incarvillateine Employing an Intramolecular Alkylation via Rh-Catalyzed Olefinic C−H Bond Activation
J. Am. Chem. Soc. 2008, 130, 6316-6317.
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187. |
Colby, D. A.; Bergman, R. G.; Ellman, J. A.
Synthesis of Dihydropyridines and Pyridines from Imines and Alkynes via C-H Activation
J. Am. Chem. Soc. 2008, 130, 3645-3651.
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186. |
Yotphan, S.; Bergman, R. G.; Ellman, J. A.
The Stereoselective Formation of Bicyclic Enamines with Bridgehead Unsaturation via Tandem C-H Bond Activation/Alkenylation/Electrocyclization
J. Am. Chem. Soc. 2008, 130, 2452-2453.
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185. |
Lewis, J. C.; Berman, A. M.; Bergman, R. G.; Ellman, J. A.
Rh(I)-Catalyzed Arylation of Heterocycles via C-H Bond Activation: Expanded Scope Through Mechanistic Insight.
J. Am. Chem. Soc. 2008, 130, 2493-2500.
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184. |
Robak, M. T.; Trincado, M.; Ellman, J. A.
Enantioselective Aza-Henry Reaction with an N-Sulfinyl Urea Organocatalyst
J. Am. Chem. Soc. 2007, 129, 15110-15111.
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183. |
Nakagawa, H.; Rech, J. C.; Sindelar, R. W.; Ellman, J. A.
Catalytic Enantioselective Addition of Arylboronic Acids to N-Boc Imines Generated in Situ
Org. Lett. 2007, 9, 5155-5157.
Write-up in Organic Process Research and Development
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182. |
Patterson, A. W.; Peltier, H. M.; Sasse, F.; Ellman, J. A.
Design, Synthesis, and Biological Properties of Highly Potent Tubulysin D Analogues
Chem. Eur. J. 2007, 13, 9534-9541.
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181. |
Tanuwidjaja, J.; Peltier, H. M.; Lewis, J. C.; Schenkel, L. B.; Ellman, J. A.
One-Pot Microwave-Promoted Synthesis of Nitriles from Aldehydes via tert-Butanesulfinyl Imines
Synthesis 2007, , 3385-3389.
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180. |
Watzke, A.; Wilson, R. M.; O’Malley, S. J.; Bergman, R. G.; Ellman, J. A.
Asymmetric Intramolecular Alkylation of Chiral Aromatic Imines via Catalytic C-H Bond Activation
Synlett 2007, , 2383-2389.
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