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229. |
Brasse, M.; Ellman, J.A.; Bergman, R.G.
A Facile, Metal- and Solvent Free, Autoxidative Coupling of Quinolines with Indoles and Pyrroles
Chem. Commun. 2011, 47, 5019-5021.
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228. |
Mahajan, S. S.; Deu, E.; Lauterwasser, E. M. W.; Leyva, M. J.; Ellman, J. A.; Bogyo, M.; Renslo, A. R.
A Fragmenting Hybrid Approach for Targeted Delivery of Multiple Therapeutic Agents to the Malaria Parasite
ChemMedChem 2011, 6, 415–419.
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227. |
Buesking, A. W.; Baguley, T. D.; Ellman, J. A.
Asymmetric Synthesis of Amines by the Knochel-Type MgCl2-Enhanced Addition of Benzyl Zinc Reagents to N-tert-Butanesulfinyl Aldimines
Org. Lett. 2011, 13, 964-967.
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226. |
Tsai, A. S.; Tauchert, M. E.; Bergman, R. G.; Ellman, J. A.
Rhodium(III)-Catalyzed Arylation of Boc-Imines via CH Bond Functionalization
J. Am. Chem. Soc. 2011, 133, 1248–1250.
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225. |
Tsai, A. S.; Brasse, M.; Bergman, R. G.; Ellman, J. A.
Rh(III)-Catalyzed Oxidative Coupling of Unactivated Alkenes via CH Activation
Org. Lett. 2011, 13, 540-542.
Research Highlight in Synfacts
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224. |
Floyd III, W. C.; Datta, G. K.; Imamura, S.; Kieler-Ferguson, H. M.; Jerger, K.; Patterson, A. W.; Fox, M. E.; Szoka, F. C.; Fréchet, J. M. J.; Ellman, J. A.
Chemotherapeutic Evaluation of a Novel Synthetic Tubulysin Analogue-Dendrimer Conjugate in C26 Tumor Bearing Mice
ChemMedChem 2011, 6, 49-53.
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223. |
Berman, A. M.; Bergman, R. G.; Ellman, J. A.
Rh(I)-Catalyzed Direct Arylation of Azines
J. Org. Chem. 2010, 75, 7863–7868.
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222. |
Crimmin, M. R.; Colby, D. A.; Bergman, R. G.; Ellman, J. A.
Synthesis and Coordination Chemistry of Tri-Substituted Benzamidrazones
J. Chem. Soc., Dalton Trans. 2011, 40, 514-522.
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221. |
Nichols, J. M.; Bishop, L. M.; Bergman, R. G.; Ellman, J. A.
Catalytic C-O Bond Cleavage of 2-Aryloxy-1-arylethanols and Its Application to the Depolymerization of Lignin Related Polymers
J. Am. Chem. Soc. 2010, 132, 12554-12555.
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220. |
Datta, G. K.; Ellman, J. A.
Racemization Free Protocol for the Synthesis of N-tert-Butanesulfinyl Ketimimes
J. Org. Chem. 2010, 75, 6283-6285.
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219. |
Leyva, M. J.; DeGiacomo, F.; Kaltenbach, L. S.; Holcomb, J.; Zhang, N.; Gafni, J.; Park, H.; Lo, D. C.; Salvesen, G. S. Ellerby, L. M.; Ellman, J. A.
Identification and Evaluation of Novel Small Molecule Pan-Caspase Inhibitors in Huntington’s Disease Models
Chem. Biol. 2010, 17, 1189-1200.
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218. |
Rawls, K. A.; Grundner, C.; Ellman, J. A.
Design and Synthesis of Novel Inhibitors for the Mycobacterium tuberculosis Phosphatase PtpB
Org. Biomol. Chem. 2010, 8, 4066-4070.
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217. |
Deu, E.; Leyva, M.; Albrow, V.; Rice, M. J.; Ellman, J. A.; Bogyo, M.
Functional studies of the Plasmodium falciparum dipeptidyl aminopeptidase I (DPAP1) using small molecule inhibitors and active site
Chem. Biol. 2010, 17, 808-819.
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216. |
Arceo, E.; Ellman, J. A.; Bergman, R. G.
Rhenium-Catalyzed Didehydroxylation of Vicinal Diols to Alkenes Using a Simple Alcohol as a Reducing Agent
J. Am. Chem. Soc. 2010, 132, 11408–11409.
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215. |
Yotphan, S.; Bergman, R. G.; Ellman, J. A.
Synthesis of Multicyclic Pyridine and Quinoline Derivatives via Intramolecular C-H Bond Functionalization
Org. Lett. 2010, 12, 2978-2981.
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214. |
Arceo, E.; Ellman, J. A.; Bergman, R. G.
A Direct, Biomass-Based Synthesis of Benzoic Acid: Formic Acid-mediated Deoxygenation of the Glucose-Derived Materials Quinic Acid and Shikimic Acid
ChemSusChem 2010, 3, 811–813.
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213. |
Robak, M. T.; Herbage, M. A.; Ellman, J. A.
Synthesis and Applications of tert-Butanesulfinamide
Chem. Rev. 2010, 110, 3600–3740 [most viewed ACS article of 2011].
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212. |
Brak, K.; Ellman, J. A.
Asymmetric Rh(I)-Catalyzed Addition of MIDA Boronates to N-tert-Butanesulfinyl Aldimines: Development and Comparison to Trifluoroborates
J. Org. Chem. 2010, 75, 3147–3150.
Research Highlight in Synfacts
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211. |
Brak, K.; Ellman, J. A.
Total Synthesis of (-)-Aurantioclavine
Org. Lett. 2010, 12, 2004–2007.
Research Highlight in Synfacts
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210. |
Brak, K.; Kerr, I. D.; Barrett, K. T.; Fuchi, N.; Debnath, M.; Ang, K.; Engel, J. C.; McKerrow, J. H.; Doyle, P. S.; Brinen, L. S.; Ellman, J. A.
Nonpeptidic Tetrafluorophenoxymethyl Ketone Cruzain Inhibitors as Promising New Leads for Chagas Disease Chemotherapy
J. Med. Chem. 2010, 53, 1763–1773.
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209. |
Drag, M.; Bogyo, M.; Ellman, J. A.; Salvesen, G. S.
Aminopeptidase Fingerprints, an Integrated Approach for Identification of Good Substrates and Optimal Inhibitors
J. Biol. Chem. 2010, 285, 3310-3318.
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208. |
Sun, C.; Su, K.-H.; Valentine, J.; Rosa-Bauza, Y. T.; Ellman, J. A.; Elboudwarej, O.; Mukherjee, B.; Craik, C. S.; Shuman, M. A.; Chen, F. F.; Zhang, X.
Time-Resolved Single-Step Protease Activity Quantification Using Nanoplasmonic Resonator Sensors
ACS Nano 2010, 4, 978–984.
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207. |
Colby, D. A.; Bergman, R. G.; Ellman, J. A.
Rhodium-Catalyzed C-C Bond Formation via Heteroatom-Directed C-H Bond Activation
Chem. Rev. 2010, 110, 624-655.
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206. |
Storgaard, M.; Ellman, J. A.
Rhodium-Catalyzed Enantioselective Addition of Arylboronic Acids to In Situ Generated N-Boc Arylimines. Preparation of (S)-tert-Butyl (4-Chlorophenyl)(Thiophen-2-yl-MethyylCarbamate
Org. Synth. 2009, 86, 360-373.
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205. |
Rawls, K. A.; Lang, T. P.; Takeuchi, J.; Imamura, S.; Baguley, T. D.; Grundner, C.; Alber, T.; Ellman, J. A.
Fragment-based discovery of selective inhibitors of the Mycobacterium tuberculosis protein tyrosine phosphatase PtpA
Bioorg. Med. Chem. Lett. 2009, 19, 6851-6854.
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204. |
Kimmel, K. L.; Robak, M. T.; Ellman, J. A.
Enantioselective Addition of Thioacetic Acid to Nitroalkenes via N-Sulfinyl Urea Organocatalysis
J. Am. Chem. Soc. 2009, 131, 8754–8755.
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203. |
Arceo, E.; Marsden, P.; Bergman, R. G.; Ellman, J. A.
An Efficient Didehydroxylation Method for the Biomass-Derived Polyols Glycerol and Erythritol. Mechanistic Studies of a Formic Acid-Mediated Deoxygenation
Chem. Commun. 2009, , 3357-3359.
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202. |
Tsai, A. S.; Wilson, R. M.; Hirada, H.; Bergman, R. G.; Ellman, J. A.
Rhodium Catalyzed Enantioselective Cylization of Substituted Imidazoles via C–H Bond Activation
Chem. Commun. 2009, , 3910-3912.
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201. |
Brak, K.; Harris, K. ; Ellman, J. A.
General One-pot Method for the Preparation of N-tert-Butanesulfinyl Amine Diastereomer Mixtures as Standards for Stereoselectivity Determinations
J. Org. Chem. 2009, 74, 3606-3608.
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200. |
Brak, K.; Ellman, J. A.
Asymmetric Synthesis of α–Branched Allylic Amines by the Rh(I)-Catalyzed Addition of Alkenyltrifluoroborates to N-tert-Butanesulfinyl Aldimines
J. Am. Chem. Soc. 2009, 131, 3850–3851.
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