Publications
| 236. |
Tauchert, M. E.; Incarvito, C. D.; Rheingold, A. L.; Bergman, R. G.; Ellman, J. A. Mechanism of the Rhodium(III)-Catalyzed Arylation of Imines via C–H Bond Functionalization: Inhibition by Substrate J. Am. Chem. Soc. 2012, 134, 1482–1485. |
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| 235. |
Kimmel, K. K.; Robak, M. T.; Thomas, S.; Lee, M. Enantio- and Diastereoselective Addition of Thioacetic Acid to Nitroalkenes via N-Sulfinyl Urea Catalysis Tetrahedron 2012, 68, 2704-2712. |
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| 234. |
Colby, D. A.; Tsai, A. S.; Bergman, R. G.; Ellman, J. A. Rhodium Catalyzed Chelation-Assisted C–H Bond Functionalization Reactions Acc. Chem. Res. 2012, 45, 814-825. |
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| 233. |
Kimmel, K.L.; Weaver, J.D.; Ellman, J.A. Enantio- and Diastereoselective Addition of Cyclohexyl Meldrum’s Acid to β- and α,β-Disubstituted Nitroalkenes via N-Sulfinyl Urea Catalysis Chem. Sci. 2012, 3, 121-125. |
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| 232. |
Hesp, K.D.; Bergman, R.G.; Ellman, J.A. Expedient Synthesis of N-Acyl Anthranilamides and β-Enamine Amides by the Rh(III)-Catalyzed Amidation of Aryl and Vinyl C-H Bonds with Isocyanates J. Am. Chem. Soc. 2011, 133, 11430–11433. |
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| 231. |
Jung, H.H.; Buesking, A.W.; Ellman, J.A. Highly Functional Group Compatible Rh-Catalyzed Addition of Arylboroxines to Activated N-tert-Butanesulfinyl Ketimines Org. Lett. 2011, 13, 3912-1915. |
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| 230. |
Robak, M.T.; Herbage, M.A.; Ellman, J.A. Development of an N-Sulfinyl Prolinamide for the Asymmetric Aldol Reaction Tetrahedron 2011, 67, 4412-4416. |
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| 229. |
Brasse, M.; Ellman, J.A.; Bergman, R.G. A Facile, Metal- and Solvent Free, Autoxidative Coupling of Quinolines with Indoles and Pyrroles Chem. Commun. 2011, 47, 5019-5021. |
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| 228. |
Mahajan, S. S.; Deu, E.; Lauterwasser, E. M. W.; Leyva, M. J.; Ellman, J. A.; Bogyo, M.; Renslo, A. R. A Fragmenting Hybrid Approach for Targeted Delivery of Multiple Therapeutic Agents to the Malaria Parasite ChemMedChem 2011, 6, 415–419. |
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| 227. |
Buesking, A. W.; Baguley, T. D.; Ellman, J. A. Asymmetric Synthesis of Amines by the Knochel-Type MgCl2-Enhanced Addition of Benzyl Zinc Reagents to N-tert-Butanesulfinyl Aldimines Org. Lett. 2011, 13, 964-967. |
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| 226. |
Tsai, A. S.; Tauchert, M. E.; Bergman, R. G.; Ellman, J. A. Rhodium(III)-Catalyzed Arylation of Boc-Imines via CH Bond Functionalization J. Am. Chem. Soc. 2011, 133, 1248–1250. |
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| 225. |
Tsai, A. S.; Brasse, M.; Bergman, R. G.; Ellman, J. A. Rh(III)-Catalyzed Oxidative Coupling of Unactivated Alkenes via CH Activation Org. Lett. 2011, 13, 540-542. Research Highlight in Synfacts |
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| 224. |
Floyd III, W. C.; Datta, G. K.; Imamura, S.; Kieler-Ferguson, H. M.; Jerger, K.; Patterson, A. W.; Fox, M. E.; Szoka, F. C.; Fréchet, J. M. J.; Ellman, J. A. Chemotherapeutic Evaluation of a Novel Synthetic Tubulysin Analogue-Dendrimer Conjugate in C26 Tumor Bearing Mice ChemMedChem 2011, 6, 49-53. |
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| 223. |
Berman, A. M.; Bergman, R. G.; Ellman, J. A. Rh(I)-Catalyzed Direct Arylation of Azines J. Org. Chem. 2010, 75, 7863–7868. |
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| 222. |
Crimmin, M. R.; Colby, D. A.; Bergman, R. G.; Ellman, J. A. Synthesis and Coordination Chemistry of Tri-Substituted Benzamidrazones J. Chem. Soc., Dalton Trans. 2011, 40, 514-522. |
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| 221. |
Nichols, J. M.; Bishop, L. M.; Bergman, R. G.; Ellman, J. A. Catalytic C-O Bond Cleavage of 2-Aryloxy-1-arylethanols and Its Application to the Depolymerization of Lignin Related Polymers J. Am. Chem. Soc. 2010, 132, 12554-12555. |
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| 220. |
Datta, G. K.; Ellman, J. A. Racemization Free Protocol for the Synthesis of N-tert-Butanesulfinyl Ketimimes J. Org. Chem. 2010, 75, 6283-6285. |
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| 219. |
Leyva, M. J.; DeGiacomo, F.; Kaltenbach, L. S.; Holcomb, J.; Zhang, N.; Gafni, J.; Park, H.; Lo, D. C.; Salvesen, G. S. Ellerby, L. M.; Ellman, J. A. Identification and Evaluation of Novel Small Molecule Pan-Caspase Inhibitors in Huntington’s Disease Models Chem. Biol. 2010, 17, 1189-1200. |
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| 218. |
Rawls, K. A.; Grundner, C.; Ellman, J. A. Design and Synthesis of Novel Inhibitors for the Mycobacterium tuberculosis Phosphatase PtpB Org. Biomol. Chem. 2010, 8, 4066-4070. |
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| 217. |
Deu, E.; Leyva, M.; Albrow, V.; Rice, M. J.; Ellman, J. A.; Bogyo, M. Functional studies of the Plasmodium falciparum dipeptidyl aminopeptidase I (DPAP1) using small molecule inhibitors and active site Chem. Biol. 2010, 17, 808-819. |
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| 216. |
Arceo, E.; Ellman, J. A.; Bergman, R. G. Rhenium-Catalyzed Didehydroxylation of Vicinal Diols to Alkenes Using a Simple Alcohol as a Reducing Agent J. Am. Chem. Soc. 2010, 132, 11408–11409. |
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| 215. |
Yotphan, S.; Bergman, R. G.; Ellman, J. A. Synthesis of Multicyclic Pyridine and Quinoline Derivatives via Intramolecular C-H Bond Functionalization Org. Lett. 2010, 12, 2978-2981. |
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| 214. |
Arceo, E.; Ellman, J. A.; Bergman, R. G. A Direct, Biomass-Based Synthesis of Benzoic Acid: Formic Acid-mediated Deoxygenation of the Glucose-Derived Materials Quinic Acid and Shikimic Acid ChemSusChem 2010, 3, 811–813. |
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| 213. |
Robak, M. T.; Herbage, M. A.; Ellman, J. A. Synthesis and Applications of tert-Butanesulfinamide Chem. Rev. 2010, 110, 3600–3740 [most viewed ACS article of 2011]. |
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| 212. |
Brak, K.; Ellman, J. A. Asymmetric Rh(I)-Catalyzed Addition of MIDA Boronates to N-tert-Butanesulfinyl Aldimines: Development and Comparison to Trifluoroborates J. Org. Chem. 2010, 75, 3147–3150. Research Highlight in Synfacts |
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| 211. |
Brak, K.; Ellman, J. A. Total Synthesis of (-)-Aurantioclavine Org. Lett. 2010, 12, 2004–2007. Research Highlight in Synfacts |
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| 210. |
Brak, K.; Kerr, I. D.; Barrett, K. T.; Fuchi, N.; Debnath, M.; Ang, K.; Engel, J. C.; McKerrow, J. H.; Doyle, P. S.; Brinen, L. S.; Ellman, J. A. Nonpeptidic Tetrafluorophenoxymethyl Ketone Cruzain Inhibitors as Promising New Leads for Chagas Disease Chemotherapy J. Med. Chem. 2010, 53, 1763–1773. |
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| 209. |
Drag, M.; Bogyo, M.; Ellman, J. A.; Salvesen, G. S. Aminopeptidase Fingerprints, an Integrated Approach for Identification of Good Substrates and Optimal Inhibitors J. Biol. Chem. 2010, 285, 3310-3318. |
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| 208. |
Sun, C.; Su, K.-H.; Valentine, J.; Rosa-Bauza, Y. T.; Ellman, J. A.; Elboudwarej, O.; Mukherjee, B.; Craik, C. S.; Shuman, M. A.; Chen, F. F.; Zhang, X. Time-Resolved Single-Step Protease Activity Quantification Using Nanoplasmonic Resonator Sensors ACS Nano 2010, 4, 978–984. |
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| 207. |
Colby, D. A.; Bergman, R. G.; Ellman, J. A. Rhodium-Catalyzed C-C Bond Formation via Heteroatom-Directed C-H Bond Activation Chem. Rev. 2010, 110, 624-655. |