Publications

252. Khan, H. A.; Ellman, J. A.
Asymmetric Synthesis of α-Aminophosphonate Esters by the Addition of Dialkyl Phosphites to tert-Butanesulfinyl Imines
Synthesis  201345, 3147–3150.
251. Lian, Y.; Hummel, J. R.; Bergman, R. G.; Ellman, J. A.
Facile Synthesis of Unsymmetrical Acridines and Phenazines by a Rhodium(III)-Catalyzed Amination, Cyclization and Aromatization Cascade
J. Am. Chem. Soc.  2013135, 12548-12551.
Research Highlight in Synfacts
250. Lian, Y.; Bergman, R. G.; Lavis, L. D.; Ellman, J. A.
Rhodium(III)-Catalyzed Indazole Synthesis by C-H Bond Functionalization and Cyclative Capture
J. Am. Chem. Soc.  2013135, 7122-7125.
249. Brasse, M.; Cámpora, J.; Begman, R. G.; Ellman, J. A.
Mechanistic Study of the Oxidative Coupling of Styrene with 2-Phenylpyridine Derivatives Catalyzed by Cationic Rhodium(III) via C–H Activation
J. Am. Chem. Soc.  2013135, 6427-6430.
248. Ischay, M. A.; Takase, M. K.; Bergman, R. G.; Ellman, J. A.
Unstabilized Azomethine Ylides for the Stereoselective synthesis of Substituted Piperidines, Tropanes and Azabicyclo[3.1.0] systems
J. Am. Chem. Soc.  2013135, 2478-2481.
Spotlights on Recent JACS Publications
247. Duttwyler, S.; Chen, S.; Takase, M. K.; Wiberg, K. B.; Bergman, R. G.; Ellman, J. A.
Proton Donor Acidity Controls Selectivity in Nonaromatic Nitrogen Heterocycle Synthesis
Science  2013339, 678-682.
C&E News Research Highlight, Write-up in Organic Process Research & Development, Research Highlight in Synfacts
246. Martin, R. M.; Bergman, R. G.; Ellman, J. A.
Synthesis of Isoquinuclidines from Highly Substituted Dihydropyridines via the Diels-Alder Reaction
Org. Lett.  201315, 444-447.
245. Lian, Y.; Huber, T.; Hesp, K. D.; Bergman, R. G.; Ellman, J. A.
Rhodium(III)-Catalyzed Alkenyl C-H Bond Functionalization: Convergent Synthesis of Furans and Pyrroles
Angew. Chem. Int. Ed.  201352, 629-633.
244. Jung, H. H.; Buesking, A. W.; Ellman, J. A.
Rh-Catalyzed Addition of Arylboroxines to Cyclic N-(Isopropanesulfinyl)ketimines
J. Org. Chem.  201277, 9593-9600.
243. Lian, Y.; Bergman, R. G.; Ellman, J. A.
Rhodium(III)-Catalyzed Synthesis of Phthalides by Cascade Addition and Cyclization of Benzimidates with Aldehydes
Chem. Sci.  20123, 3088-3092.
242. Verdoes, M.; Edgington, L. E.; Scheeren, F. A.; Leyva, M.; Blum, G.; Weiskopf, K.; Bachmann, M. H.; Ellman, J. A.; Bogyo, M.
A Nonpeptidic Cathepsin S Activity-Based Probe for Noninvasive Optical Imaging of Tumor-Associated Macrophages
Chem. Biol.  201219, 619-628.
241. Kimmel, K. L.; Weaver, J. D.; Lee, M.; Ellman, J. A.
Enantio- and Diastereoselective Addition of Cyclohexyl Meldrum’s Acid to β- and α,β-Disubstituted Nitroalkenes via N-Sulfinyl Urea Catalysis
J. Am. Chem. Soc.  2012134, 9058-9061.
Research Highlight in Synfacts
240. Xue, Y.; Chowdhury, S.; Liu, X.; Akiyama, Y.; Ellman, J. A.; Ha, Y.
Conformational Change in Rhomboid Protease GlpG Induced by Inhibitor Binding to Its S′ Subsites
Biochemistry  201251, 3723-3731.
239. Hesp, K. D.; Bergman, R. G.; Ellman, J. A.
Rhodium-Catalyzed Synthesis of Branched Amines by Direct Addition of Benzamides to Imines
Org. Lett.   201214, 2304-2307.
External Link
238. Martin, R. M.; Bergman, R. G.; Ellman, J. A.
Synthesis of Pyridines from Ketoximes and Terminal Alkynes via C–H Bond Functionalization
J. Org. Chem.  201277, 2501–2507.
Research Highlight in Synfacts
237. Duttwyler, S.; Rheingold, A. L.; Bergman, R. G.; Ellman, J. A.
Highly Diastereoselective Synthesis of Tetrahydropyridines by a C–H Activation–Cyclization–Reduction Cascade
J. Am. Chem. Soc.  2012134, 4064-4067.
Research Highlight in Synfacts
236. Tauchert, M. E.; Incarvito, C. D.; Rheingold, A. L.; Bergman, R. G.; Ellman, J. A.
Mechanism of the Rhodium(III)-Catalyzed Arylation of Imines via C–H Bond Functionalization: Inhibition by Substrate
J. Am. Chem. Soc.  2012134, 1482–1485.
235. Kimmel, K. K.; Robak, M. T.; Thomas, S.; Lee, M.
Enantio- and Diastereoselective Addition of Thioacetic Acid to Nitroalkenes via N-Sulfinyl Urea Catalysis
Tetrahedron  201268, 2704-2712.
234. Colby, D. A.; Tsai, A. S.; Bergman, R. G.; Ellman, J. A.
Rhodium Catalyzed Chelation-Assisted C–H Bond Functionalization Reactions
Acc. Chem. Res.  201245,  814-825.
233. Kimmel, K.L.; Weaver, J.D.; Ellman, J.A.
Enantio- and Diastereoselective Addition of Cyclohexyl Meldrum’s Acid to β- and α,β-Disubstituted Nitroalkenes via N-Sulfinyl Urea Catalysis
Chem. Sci.  20123, 121-125.
232. Hesp, K.D.; Bergman, R.G.; Ellman, J.A.
Expedient Synthesis of N-Acyl Anthranilamides and β-Enamine Amides by the Rh(III)-Catalyzed Amidation of Aryl and Vinyl C-H Bonds with Isocyanates
J. Am. Chem. Soc.  2011133, 11430–11433.
231. Jung, H.H.; Buesking, A.W.; Ellman, J.A.
Highly Functional Group Compatible Rh-Catalyzed Addition of Arylboroxines to Activated N-tert-Butanesulfinyl Ketimines
Org. Lett.  201113, 3912-1915.
230. Robak, M.T.; Herbage, M.A.; Ellman, J.A.
Development of an N-Sulfinyl Prolinamide for the Asymmetric Aldol Reaction
Tetrahedron  201167, 4412-4416.
229. Brasse, M.; Ellman, J.A.; Bergman, R.G.
A Facile, Metal- and Solvent Free, Autoxidative Coupling of Quinolines with Indoles and Pyrroles
Chem. Commun.   201147, 5019-5021.
228. Mahajan, S. S.; Deu, E.; Lauterwasser, E. M. W.; Leyva, M. J.; Ellman, J. A.; Bogyo, M.; Renslo, A. R.
A Fragmenting Hybrid Approach for Targeted Delivery of Multiple Therapeutic Agents to the Malaria Parasite
ChemMedChem  20116, 415–419.
227. Buesking, A. W.; Baguley, T. D.; Ellman, J. A.
Asymmetric Synthesis of Amines by the Knochel-Type MgCl2-Enhanced Addition of Benzyl Zinc Reagents to N-tert-Butanesulfinyl Aldimines
Org. Lett.   201113, 964-967.
226. Tsai, A. S.; Tauchert, M. E.; Bergman, R. G.; Ellman, J. A.
Rhodium(III)-Catalyzed Arylation of Boc-Imines via CH Bond Functionalization
J. Am. Chem. Soc.  2011133, 1248–1250.
225. Tsai, A. S.; Brasse, M.; Bergman, R. G.; Ellman, J. A.
Rh(III)-Catalyzed Oxidative Coupling of Unactivated Alkenes via CH Activation
Org. Lett.  201113, 540-542.
Research Highlight in Synfacts
224. Floyd III, W. C.; Datta, G. K.; Imamura, S.; Kieler-Ferguson, H. M.; Jerger, K.; Patterson, A. W.; Fox, M. E.; Szoka, F. C.; Fréchet, J. M. J.; Ellman, J. A.
Chemotherapeutic Evaluation of a Novel Synthetic Tubulysin Analogue-Dendrimer Conjugate in C26 Tumor Bearing Mice
ChemMedChem  20116,  49-53.
223. Berman, A. M.; Bergman, R. G.; Ellman, J. A.
Rh(I)-Catalyzed Direct Arylation of Azines
J. Org. Chem.  201075, 7863–7868.

Pages