Publications
290. |
Potter, T. J.; Kamber, D. N.; Mercado, B. Q.; Ellman, J. A. Rh(III)-Catalyzed Aryl and Alkenyl C–H Bond Addition to Diverse Nitroalkenes ACS Catal. 2017, 7, 150–153. |
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289. |
Hummel, J. R.; Ellman, J. A. Convergent Synthesis of α-Branched Amines by Transition-Metal-Catalyzed C−H Bond Additions to Imines Isr. J. Chem. 2017, 57, 916–931 [honoring Bob Bergman's Wolf Prize]. |
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288. |
Wangweerawong, A.; Kolmar. S.; Ellman, J. A. Preparation of (S)-Nonafluorobutanesulfinamide Org. Synth. 2016, 93, 319-330. |
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287. |
Chen, S.; Bacauanu, V.; Knecht, T.; Mercado, B. Q.; Bergman, R. G.; Ellman, J. A. New Regio- and Stereoselective Cascades via Unstabilized Azomethine Ylide Cycloadditions for the Synthesis of Highly Substituted Tropane and Indolizidine Frameworks J. Am. Chem. Soc. 2016, 138, 12664–12670. |
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286. |
Potter, T. J.; Ellman, J. A. Rh(III)-Catalyzed C–H Bond Addition/Amine-Mediated Cyclization of Bis-Michael Acceptors Org. Lett. 2016, 18, 3838–3841. |
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285. |
Jamali, H.; Khan, H. A.; Tjin, C. C.; Ellman, J. A. Cellular Activity of New Small Molecule Protein Arginine Deiminase 3 (PAD3) Inhibitors ACS Med. Chem. Lett. 2016, 7, 847–851. |
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284. |
Weinstein, A. B.; Ellman, J. A. Convergent Synthesis of Diverse Nitrogen Heterocycles via Rh(III)-Catalyzed C–H Conjugate Addition/Cyclization Reactions Org. Lett. 2016, 18, 3294-3297. Research Highlight in Synfacts |
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283. |
Boerth, J. A.; Hummel, J. R.; Ellman, J. A. Highly Stereoselective Cobalt(III)-Catalyzed Three-Component C−H Bond Addition Cascade Angew. Chem. Int. Ed. 2016, 55, 12650-12654 [Hot Paper]. Write-up in Organic Process Research & Development, Research Highlight in Synfacts |
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282. |
Phelan, J. P.; Ellman, J. A. Conjugate Addition–Enantioselective Protonation Reactions Beilstein J. Org. Chem. 2016, 12, 1203–1228. |
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281. |
Mesganaw, T.; Elman, J. A. 4-(Diethylphosphino)-N,N-dimethylaniline e-EROS Encyclopedia of Reagents for Organic Synthesis 2016, , . |
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280. |
Phelan, J. P.; Ellman, J. A. Catalytic Enantioselective Addition of Pyrazol-5-ones to Trisubstituted Nitroalkenes with an N-Sulfinylurea Organocatalyst Adv. Synth. Catal. 2016, 358, 1713–1718. |
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279. |
Wangweerawong, A.; Hummel, J. R.; Bergman, R. G.; Ellman, J. A. Preparation of Enantiomerically Pure Perfluorobutanesulfinamide and Its Application to the Asymmetric Synthesis of α-Amino Acids J. Org. Chem. 2016, 81, 1547–1557. |
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278. |
Boerth, J. A.; Ellman, J. A. Rh(III)-Catalyzed Diastereoselective C–H Bond Addition/Cyclization Cascade of Enone Tethered Aldehydes Chem. Sci. 2016, 7, 1474-1479. |
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277. |
Xu, J.; Kurup, P.; Baguley, T.; Foscue, E.; Ellman J. A.; Nairn, A. C.; Lombroso, P. J. Inhibition of the Tyrosine Phosphatase STEP61 Restores BDNF Expression and Reverses Motor and Cognitive Deficits in Phencyclidine-Treated Mice Cell. Mol. Life Sci. 2016, 73, 1503-1514. |
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276. |
Azkona, G.; Saavedra, A.; Aira, Z.; Aluja, D.; Xifró, X.; Baguley, T.; Alberch, J.; Ellman J. A.; Lombroso, P. J.; Azkue, J. J.; Pérez-Navarro, E. Striatal-Enriched Protein Tyrosine Phosphatase Modulates Nociception: Evidence from Genetic Deletion and Pharmacological Inhibition Pain 2016, 157, 377-86. |
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275. |
Xu, J.; Kurup, P. K.; Azkona, G. M.; Baguley, T. D.; Saavedra, A. C.; Nairn, A. C.; Ellman, J. A.; Perez-Navarro, E.; Lombroso, P. A. Down-Regulation of BDNF in Cell and Animal Models Increases Striatal-Enriched Protein Tyrosine Phosphatase STEP61 Levels J. Neurochem. 2016, 136, 285–294. |
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274. |
Phillips, E. M.; Mesganaw, T.; Patel, A. Duttwyler, S.; Mercado, B. Q.; Houk, K. N.; Ellman, J. A. Synthesis of ent-Ketorfanol via a C–H Alkenylation/ Torquoselective 6π-Electrocyclization Cascade Angew. Chem. Int. Ed. 2015, 54, 12044–12048. Research Highlight in Synfacts |
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273. |
Neitz, R. J.; Bryant, C.; Chen, S.; Gut, J.; Caselli, E. H.; Ponce, S.; Chowdhury, S.; Xu, H.; Arkin, M. R.; Ellman, J. A.; Renslo, A. R. Tetrafluorophenoxymethyl Ketone Cruzain Inhibitors with Improved Pharmacokinetic Properties as Therapeutic Leads for Chagas’ Disease Bioorg. Med. Chem. Lett. 2015, 25, 4834–4837. |
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272. |
Chen, S.; Mercado, B. Q.; Bergman, R. G.; Ellman, J. A. Regio- and Diastereoselective Synthesis of Highly Substituted, Oxygenated Piperidines from Tetrahydropyridines J. Org. Chem. 2015, 80, 6660–6668. |
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271. |
Chen, S.; Bergman, R. G.; Ellman, J. A. Facile Rh(III)-Catalyzed Synthesis of Fluorinated Pyridines Org. Lett. 2015, 17, 2567–2569. |
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270. |
Hummel, J. R.; Ellman, J. A. Cobalt(III)-Catalyzed C–H Bond Amidation with Isocyanates Org. Lett. 2015, 17, 2400–2403. |
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269. |
Oresic Bender, K.; Ofori, L.; van der Linden, W. A.; Mock, E. D.; Datta, G.; Chowdhury, S.; Li, H.; Segal, E.; Lopez, M. S.; Ellman, J. A.; Figdor, C. G.; Bogyo, M.; Verdoes, M. Design of a Highly Selective Quenched Activity-Based Probe and Its Application in Dual Color Imaging Studies of Cathepsin S Activity Localization J. Am. Chem. Soc. 2015, 137, 4771–4777. |
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268. |
Jamali, H.; Khan, H. A.; Stringer, J. A.; Chowdhury, S. Ellman, J. A. Identification of Multiple Structurally-Distinct, Nonpeptidic Small Molecule Inhibitors of Protein Arginine Deiminase 3 Using a Substrate-Based Fragment Method J. Am. Chem. Soc. 2015, 137, 3616–3621. |
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267. |
Otley, K. D.; Ellman, J. A. An Efficient Method for the Preparation of Styrene Derivatives via Rh(III)-Catalyzed Direct C–H Vinylation Org. Lett. 2015, 17, 1332–1335 [ACS Select Virtual Issue on C-H Functionalization]. |
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266. |
Matsushima, Y.; Phillips, E. M.; Bergman, R. G.; Ellman, J. A. Rh(I)-Catalyzed Cycloisomerization of 1,6-Enynes Synlett 2015, 26, 1533–1536. |
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265. |
Baguley, T. D.; Nairn, A. C.; Lombroso, P. J.; Ellman, J. A. Synthesis of Benzopentathiepin Analogs and Their Evaluation as Inhibitors of the Phosphatase STEP Bioorg. Med. Chem. Lett. 2015, 25, 1050-1052. |
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264. |
Hummel, J. R.; Ellman, J. A. Cobalt(III)-Catalyzed Synthesis of Indazoles and Furans by C–H Bond Functionalization/Addition/Cyclization Cascades J. Am. Chem. Soc. 2015, 137, 490–498. Write-up in Organic Process Research and Development |
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263. |
Otley, K. D.; Ellman, J. A. A Lewis Acid-Catalyzed Annulation to 2,1-Benzisoxazoles J. Org. Chem. 2014, 79, 8296–8303. |
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262. |
Mesganaw, T.; Ellman, J. A. Convergent Synthesis of Diverse Tetrahydropyridines via Rh(I)-Catalyzed C–H Functionalization Sequences Org. Process Res. Dev. 2014, 18, 1097–1104. |
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261. |
Mesganaw, T.; Ellman, J. A. Preparative Synthesis of Highly Substituted Tetrahydropyridines via a Rh(I)-Catalyzed C–H Functionalization Sequence Org. Process Res. Dev. 2014, 18, 1105–1109. |