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295. |
Boerth, J. A.; Ellman, J. A.
A Convergent Synthesis of Functionalized Alkenyl Halides via Co(III)-Catalyzed Three-Component C-H Bond Addition
Angew. Chem. Int. Ed. 2017, 56, 9976–9980 [Very Important Paper].
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294. |
Halskov, K.; Roth, H.; Ellman, J. A.
Synthesis of [5,6]-Bicyclic Heterocycles with a Ring-Junction Nitrogen via Rh(III)-Catalyzed C-H Functionalization of Alkenyl Azoles
Angew. Chem. Int. Ed. 2017, 56, 9183–9187.
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293. |
Potter, T. J.; Ellman, J. A.
Total Synthesis of (+)-Pancratistatin by the Rh(III)-Catalyzed Addition of a Densely Functionalized Benzamide to a Sugar-Derived Nitroalkene
Org. Lett. 2017, 19, 2985–2988.
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292. |
Tran, G.; Hesp, K. D.; Mascitti, V.; Ellman, J. A.
Base-Controlled Completely Selective Linear or Branched Rhodium(I)-Catalyzed C−H ortho-Alkylation of Azines without Preactivation
Angew. Chem. Int. Ed. 2017, 56, 5899–5903.
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291. |
Hummel, J. R.; Boerth, J. A.; Ellman, J. A.
Transition-Metal-Catalyzed C–H Bond Addition to Carbonyls, Imines, and Related Polarized π Bonds
Chem. Rev. 2017, 117, 9163–9227.
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290. |
Potter, T. J.; Kamber, D. N.; Mercado, B. Q.; Ellman, J. A.
Rh(III)-Catalyzed Aryl and Alkenyl C–H Bond Addition to Diverse Nitroalkenes
ACS Catal. 2017, 7, 150–153.
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289. |
Hummel, J. R.; Ellman, J. A.
Convergent Synthesis of α-Branched Amines by Transition-Metal-Catalyzed C−H Bond Additions to Imines
Isr. J. Chem. 2017, 57, 916–931 [honoring Bob Bergman's Wolf Prize].
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288. |
Wangweerawong, A.; Kolmar. S.; Ellman, J. A.
Preparation of (S)-Nonafluorobutanesulfinamide
Org. Synth. 2016, 93, 319-330.
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287. |
Chen, S.; Bacauanu, V.; Knecht, T.; Mercado, B. Q.; Bergman, R. G.; Ellman, J. A.
New Regio- and Stereoselective Cascades via Unstabilized Azomethine Ylide Cycloadditions for the Synthesis of Highly Substituted Tropane and Indolizidine Frameworks
J. Am. Chem. Soc. 2016, 138, 12664–12670.
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286. |
Potter, T. J.; Ellman, J. A.
Rh(III)-Catalyzed C–H Bond Addition/Amine-Mediated Cyclization of Bis-Michael Acceptors
Org. Lett. 2016, 18, 3838–3841.
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285. |
Jamali, H.; Khan, H. A.; Tjin, C. C.; Ellman, J. A.
Cellular Activity of New Small Molecule Protein Arginine Deiminase 3 (PAD3) Inhibitors
ACS Med. Chem. Lett. 2016, 7, 847–851.
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284. |
Weinstein, A. B.; Ellman, J. A.
Convergent Synthesis of Diverse Nitrogen Heterocycles via Rh(III)-Catalyzed C–H Conjugate Addition/Cyclization Reactions
Org. Lett. 2016, 18, 3294-3297.
Research Highlight in Synfacts
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283. |
Boerth, J. A.; Hummel, J. R.; Ellman, J. A.
Highly Stereoselective Cobalt(III)-Catalyzed Three-Component C−H Bond Addition Cascade
Angew. Chem. Int. Ed. 2016, 55, 12650-12654 [Hot Paper].
Write-up in Organic Process Research & Development, Research Highlight in Synfacts
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282. |
Phelan, J. P.; Ellman, J. A.
Conjugate Addition–Enantioselective Protonation Reactions
Beilstein J. Org. Chem. 2016, 12, 1203–1228.
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281. |
Mesganaw, T.; Elman, J. A.
4-(Diethylphosphino)-N,N-dimethylaniline
e-EROS Encyclopedia of Reagents for Organic Synthesis 2016, , .
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280. |
Phelan, J. P.; Ellman, J. A.
Catalytic Enantioselective Addition of Pyrazol-5-ones to Trisubstituted Nitroalkenes with an N-Sulfinylurea Organocatalyst
Adv. Synth. Catal. 2016, 358, 1713–1718.
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279. |
Wangweerawong, A.; Hummel, J. R.; Bergman, R. G.; Ellman, J. A.
Preparation of Enantiomerically Pure Perfluorobutanesulfinamide and Its Application to the Asymmetric Synthesis of α-Amino Acids
J. Org. Chem. 2016, 81, 1547–1557.
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278. |
Boerth, J. A.; Ellman, J. A.
Rh(III)-Catalyzed Diastereoselective C–H Bond Addition/Cyclization Cascade of Enone Tethered Aldehydes
Chem. Sci. 2016, 7, 1474-1479.
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277. |
Xu, J.; Kurup, P.; Baguley, T.; Foscue, E.; Ellman J. A.; Nairn, A. C.; Lombroso, P. J.
Inhibition of the Tyrosine Phosphatase STEP61 Restores BDNF Expression and Reverses Motor and Cognitive Deficits in Phencyclidine-Treated Mice
Cell. Mol. Life Sci. 2016, 73, 1503-1514.
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276. |
Azkona, G.; Saavedra, A.; Aira, Z.; Aluja, D.; Xifró, X.; Baguley, T.; Alberch, J.; Ellman J. A.; Lombroso, P. J.; Azkue, J. J.; Pérez-Navarro, E.
Striatal-Enriched Protein Tyrosine Phosphatase Modulates Nociception: Evidence from Genetic Deletion and Pharmacological Inhibition
Pain 2016, 157, 377-86.
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275. |
Xu, J.; Kurup, P. K.; Azkona, G. M.; Baguley, T. D.; Saavedra, A. C.; Nairn, A. C.; Ellman, J. A.; Perez-Navarro, E.; Lombroso, P. A.
Down-Regulation of BDNF in Cell and Animal Models Increases Striatal-Enriched Protein Tyrosine Phosphatase STEP61 Levels
J. Neurochem. 2016, 136, 285–294.
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274. |
Phillips, E. M.; Mesganaw, T.; Patel, A. Duttwyler, S.; Mercado, B. Q.; Houk, K. N.; Ellman, J. A.
Synthesis of ent-Ketorfanol via a C–H Alkenylation/ Torquoselective 6π-Electrocyclization Cascade
Angew. Chem. Int. Ed. 2015, 54, 12044–12048.
Research Highlight in Synfacts
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273. |
Neitz, R. J.; Bryant, C.; Chen, S.; Gut, J.; Caselli, E. H.; Ponce, S.; Chowdhury, S.; Xu, H.; Arkin, M. R.; Ellman, J. A.; Renslo, A. R.
Tetrafluorophenoxymethyl Ketone Cruzain Inhibitors with Improved Pharmacokinetic Properties as Therapeutic Leads for Chagas’ Disease
Bioorg. Med. Chem. Lett. 2015, 25, 4834–4837.
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272. |
Chen, S.; Mercado, B. Q.; Bergman, R. G.; Ellman, J. A.
Regio- and Diastereoselective Synthesis of Highly Substituted, Oxygenated Piperidines from Tetrahydropyridines
J. Org. Chem. 2015, 80, 6660–6668.
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271. |
Chen, S.; Bergman, R. G.; Ellman, J. A.
Facile Rh(III)-Catalyzed Synthesis of Fluorinated Pyridines
Org. Lett. 2015, 17, 2567–2569.
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270. |
Hummel, J. R.; Ellman, J. A.
Cobalt(III)-Catalyzed C–H Bond Amidation with Isocyanates
Org. Lett. 2015, 17, 2400–2403.
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269. |
Oresic Bender, K.; Ofori, L.; van der Linden, W. A.; Mock, E. D.; Datta, G.; Chowdhury, S.; Li, H.; Segal, E.; Lopez, M. S.; Ellman, J. A.; Figdor, C. G.; Bogyo, M.; Verdoes, M.
Design of a Highly Selective Quenched Activity-Based Probe and Its Application in Dual Color Imaging Studies of Cathepsin S Activity Localization
J. Am. Chem. Soc. 2015, 137, 4771–4777.
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268. |
Jamali, H.; Khan, H. A.; Stringer, J. A.; Chowdhury, S. Ellman, J. A.
Identification of Multiple Structurally-Distinct, Nonpeptidic Small Molecule Inhibitors of Protein Arginine Deiminase 3 Using a Substrate-Based Fragment Method
J. Am. Chem. Soc. 2015, 137, 3616–3621.
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267. |
Otley, K. D.; Ellman, J. A.
An Efficient Method for the Preparation of Styrene Derivatives via Rh(III)-Catalyzed Direct C–H Vinylation
Org. Lett. 2015, 17, 1332–1335 [ACS Select Virtual Issue on C-H Functionalization].
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266. |
Matsushima, Y.; Phillips, E. M.; Bergman, R. G.; Ellman, J. A.
Rh(I)-Catalyzed Cycloisomerization of 1,6-Enynes
Synlett 2015, 26, 1533–1536.
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