Publications

132. Schenkel, L. B.; Ellman, J. A.
Application of P,N-Sulfinyl Imine Ligands to Iridium-Catalyzed Asymmetric Hydrogenation of Olefins
J. Org. Chem.  2004, 69, 1800-1802.
131. Lewis, J. C. Wiedemann, S. H.; Bergman, R. G.; Ellman, J. A.
Arylation of Heterocycles via Rhodium-Catalyzed C-H Bond Functionalization
Org. Lett.  2004, 6, 35-38.
130. Evans, J. W.; Ellman, J. A.
Stereoselective Synthesis of 1,2-Disubstituted beta-Amino Alcohols by Nucleophilic Addition to N-tert-Butanesulfinyl aldimines
J. Org. Chem.  2003, 68, 9948-9957.
129. Wood, W.; Huang, L.; Ellman, J. A.
Synthesis of a Diverse Library of Mechanism-Based Cysteine Protease Inhibitors
J. Comb. Chem.  2003, 5, 869-880.
128. Boitano, A.; Ellman, J. A.; Glick, G. D.; Opipari, A. W.
The Proapoptotic Benzodiazepine BZ-423 Affects the Growth and Survival of Malignant B Cells
Cancer Res.  2003, 63, 6870-6876.
http://cancerres.aacrjournals.org/content/63/20/6870.full
127. Boitano, A.; Leonetii, F.; Emal, C.; Ellman, J. A.; Roush, W. R.; Opipari, A. W.; Glick, G. D.
Structure Activity Studies of a Novel Cytotoxic Benzodiazepine
Bioorg. Med. Chem. Lett.  2003, 13, 3327-3330.
126. Kochi, T.; Tang, T. P.; Ellman, J. A.
Development and Application of a New General Method for the Asymmetric Synthesis of syn- and anti-1,3-Amino Alcohols
J. Am. Chem. Soc.  2003, 125, 11276-11282.
125. Jain, R. K.; Trias, J.; Ellman, J. A.
D-Ala-D-Lac Binding is Not Required for the High Activity of Vancomycin Dimers Against Vancomycin Resistant Enterococci
J. Am. Chem. Soc.  2003, 125, 8740-8741.
124. Mukade, T.; Dragoli, D. R.; Ellman, J. A.
Parallel Solution-Phase Asymmetric Synthesis of alpha-Branched Amines
J. Comb. Chem.  2003, 5, 590-596.
123. Tan, K. L.; Vasudevan, A.; Bergman, R. G.; Ellman, J. A.; Souers, A. J.
Microwave Assisted C-H Bond Activation: A Rapid Entry into Functionalized Heterocycles
Org. Lett.  2003, 5, 2131-2134.
122. Ahrendt, K. A.; Bergman, R. G.; Ellman, J. A
Synthesis of a Tricyclic Mescaline Analog by Catalytic C-H Bond Activation
Org. Lett.  2003, 5, 1301-1303.
121. Weix, D. J.; Ellman, J. A.
An Improved Synthesis of tert-Butanesulfinamide Suitable for Large Scale Production
Org. Lett.  2003, 5, 1317-1320.
120. Leiting, B.; Pryor, K. D.; Wu, J. K.; Marsilio, F.; Patel, R. A.; Craik, C. S.; Ellman, J. A.; Cummings, R. T.; Thornberry, N.
Catalytic Properties and Inhibition of Proline-Specific Dipeptidyl Peptidases II, IV and VII
Biochem. J.  2003, 371, 525-532.
119. Ahrendt, K. A.; Olsen, J. A.; Wakao, M.; Trias, J. Ellman, J. A.
Identification of Potent and Broad-Spectrum Antibiotics from SAR Studies of a Synthetic Vancomycin Analog
Bioorg. Med. Chem. Lett.  2003, 13, 1683-1686.
118. Cawley, N. X.; Chino, M.; Maldonado, A.; Rodriguez, Y. M.; Loh, Y. P.; Ellman, J. A.
Synthesis and Characterization of the First Potent Inhibitor of Yapsin 1. Implications for the Study of Yapsin-Like Enzymes
J. Biol. Chem.  2003, 278, 5523-5530.
117. Asojo, O. A.; Gulnik. S. V.; Afonina, E.; Yu, B.; Ellman, J. A.; Haque, T. S.; Silva, A. M.
Novel Uncomplexed and Complexed Structures of Plasmepsin II, an Aspartic Protease from Plasmodium falciparum
J. Mol. Biol.  2003, 327, 173-181.
116. Schenkel, L. B.; Ellman, J. A.
Novel Sulfinyl Imine Ligands for Asymmetric Catalysis
Org. Lett.  2003, 5, 545-548.
115. Bednarski, J. J.; Warner, R. E.; Rao, T.; Leonetti, F.; Yung, R.; Richardson, B. C.; Johnson, K. J.; Ellman, J. A. Opipari, A. W.; Glick, G. D.
Attenuation of Autoimmune Disease in Fas-Deficient Mice by Treatment with a Cytotoxic Benzodiazepine
Arthritis & Rheumatism  2003, 48, 757-766.
114. Huang, L.; Brinen, L. S.; Ellman, J. A.
Crystal Structures of Reversible Ketone-Based Inhibitors of the Cysteine Protease Cruzain
Bioorg. Med. Chem.  2003, 11, 21-29.
113. Ellman, J. A.
Applications of tert-Butanesulfinamide in the Asymmetric Synthesis of Amines
Pure Appl. Chem.  2003, 75, 39-46.
112. Owens, T. D.; Souers, A. J.; Ellman, J. A.
The Preparation and Utility of Bis(sulfinyl)imidoamidine Ligands for the Copper-Catalyzed Diels Alder Reaction
J. Org. Chem.  2003, 68, 3-10.
111. Blum, S. A.; Bergman, R. G.; Ellman, J. A.
Enantioselective Oxidation of Di-tert-Butyl Disulfide with a Vanadium Catalyst: Progress toward Mechanism Elucidation
J. Org. Chem.  2003, 68, 150-155.
110. Salisbury, C. M.; Maly, D. J.; Ellman, J. A.
Peptide Microarrays for the Determination of Substrate Specificity
J. Am. Chem. Soc.  2002, 124, 14868-14870.
109. Ellman, J. A.; Owens, T. D.; Tang, T. P.
N-tert-Butanesulfinyl Imines: Versatile Intermediates for the Asymmetric Synthesis of Amines
Acc. Chem. Res.  2002, 35, 984-995.
108. Tang, T. P.; Ellman, J. A.
Asymmetric Synthesis of beta-Amino Acid Derivatives Incorporating a Broad Range of Substitution Patterns by Enolate Additions to tert-Butanesulfinyl Imines
J. Org. Chem.  2002, 67, 7819-7832.
107. Blatt, N. B.; Bednarski, J. J.; Warner, R. E.; Leonetti, F.; Johnson, K. M.; Boitano, A.; Yung, R.; Richardson, B. C.; Johnson, K. J.; Ellman, J. A. Opipari, A. W.; Glick, G. D.
Benzodiazepine-Induced Superoxide Signals B Cell Apoptosis: Mechanistic Insight and Potential Therapeutic Utility
J. Clin. Invest.  2002, 110, 1123-1132.
106. Tan, K. L.; Bergman, R. G.; Ellman, J. A.
Intermolecular Coupling of Alkenes to Heterocycles via Rhodium-Catalyzed C-H Bond Activation
J. Am. Chem. Soc.  2002, 124, 13964-13965.
105. Huang, L.; Ellman, J. A.
General Solid-Phase Procedure to Prepare Novel Cyclic Ketone Inhibitors of the Cysteine Protease Cruzain
Bioorg. Med. Chem. Lett.  2002, 12, 2993-2996.
104. Choi, C. Y. H.; Schneider, E. L.; Kim, J. M.; Gluzman, I. Y.; Goldberg, D. E.; Ellman, J. A.; Marletta, A.
Interference with Heme Binding to Histidine-Rich Protein-2 As an Antimalarial Strategy
Chem. Biol.  2002, 9, 881-889.
103. Chino, M.; Wakao, M.; Ellman, J. A.
Efficient Method to Prepare Hydroxyethylamine-Based Aspartyl Protease Inhibitors with Diverse P1 Side Chains
Tetrahedron  2002, 58, 6305-6310.

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