Publications

320. Confair, D. N.; Greenwood, N. S.; Mercado, B. Q.; Ellman, J. A.
Rh(III)-Catalyzed Imidoyl C–H Carbamylation and Cyclization to Bicyclic [1,3,5]Triazinones
Org. Lett.   202022, ASAP.
319. Dongbang, S.; Ellman, Jonathan A.
Synthesis of Nitrile Bearing Acyclic Quaternary Centers via Co(III)‐Catalyzed Sequential C–H Bond Addition to Dienes and N‐Cyanosuccinimide
Angew. Chem. Int. Ed.  202059, Early View.
318. Gannam, Z. T. K.; Min, K.; Shillingford, S. R.; Zhang, L.; Herrington, J.; Abriola, L.; Gareiss, P. C.; Pantouris, G.; Tzouvelekis, A.; et al.
An allosteric site on MKP5 reveals a strategy for small molecule inhibition
Science Signaling  202013, eaba3043.
317. Walker, M. M.; Koronkiewicz, B.; Chen, S.; Houk, K. N.; Mayer, J. M.; Ellman, J. A.
Highly Diastereoselective Functionalization of Piperidines by Photoredox Catalyzed α-Amino C–H Arylation and Epimerization
J. Am. Chem. Soc.  2020142, 8194-8202 [ChemRxiv, 2019: doi.org/10.26434/chemrxiv.11336642.v1].
Research Highlight in Synfacts, Featured in Org. Chem. Highlights: C-N Ring Construction
316. Streit, A. D.; Zoll, A. J.; Hoang, G. L.; Ellman, J. A.
Annulation of Hydrazones and Alkynes via Rhodium(III)-Catalyzed Dual C–H Activation: Synthesis of Pyrrolopyridazines and Azolopyridazines
Org. Lett.  202022, 1217-1221.
315. Shen, Z.; Li, C.; Mercado, B. Q.; Ellman, J. A.
Cobalt(III)-Catalyzed Diastereoselective Three-Component C–H Bond Addition to Butadiene and Activated Ketones
Synthesis  202052, 1239-1246 [Domino C–H functionalization reaction/cascade catalysis in honor of Prof. Mark Lautens].
314. Scamp, R. J.; deRamon, E.; Paulson, E. K.; Miller, S. J.; Ellman, J. A.
Co(III)-Catalyzed C-H Amidation of Dehydroalanine for the Site-Selective Structural Diversification of Thiostrepton
Angew. Chem. Int. Ed.  202059, 890-895.
313. Ellman, J. A.; Ackermann, L.; Shi, B.-F.
The Breadth and Depth of C–H Functionalization
J. Org. Chem.  201984, 12701-12704.
312. Maity, S.; Potter, T. J.; Ellman, J. A.
α-Branched Amines by Catalytic 1,1-Addition of C–H Bonds and Aminating Agents to Terminal Alkenes
Nat. Catal.  20192, 756–762.
311. Dongbang, S.; Shen, Z.; Ellman, J. A.
Synthesis of Homoallylic Alcohols with Acyclic Quaternary Centers via CoIII‐Catalyzed Three‐Component C–H Bond Addition to Internally Substituted Dienes and Carbonyls
Angew. Chem. Int. Ed.  201958, 12590–12594 [Hot Paper].
310. Hoang, G. L.; Zoll, A. J.; Ellman, J. A.
Three-Component Coupling of Aldehydes, 2-Aminopyridines, and Diazo Esters via Rhodium(III)-Catalyzed Imidoyl C–H Activation: Synthesis of Pyrido[1,2-a]pyrimidin-4-ones
Org. Lett.  201921, 3886-3890 [cover picture for issue 11, June 7].
Write-up in Organic Process Research and Development
309. Chen, S.; Chan, A. Y.; Walker, M. M.; Ellman, J. A.; Houk, K. N.
π-Facial Selectivities in Hydride Reductions of Hindered Endocyclic Iminium Ions
J. Org. Chem.  201984, 273–281.
308. Dongbang, S.; Pedersen, B.; Ellman, J. A.
Asymmetric Synthesis of (−)-Naltrexone
Chem. Sci.  201910, 535–541 [Editor's Choice].
307. Hoang, G. L.; Streit, A. D.; Ellman, J. A.
Three-Component Coupling of Aldehydes, Aminopyrazoles, and Sulfoxonium Ylides via Rhodium(III)-Catalyzed Imidoyl C–H Activation: Synthesis of Pyrazolo[1,5-a]pyrimidines
J. Org. Chem.  201883, 15347-15360.
Sigma/Aldrich technology spotlight and commercial availability of ketosulfoxonium ylides
306. Chandra Tjin, C.; Wissner, R.; Jamali, H.; Schepartz, A.; Ellman, J. A.
Synthesis and Biological Evaluation of an Indazole-Based Selective Protein Arginine Deiminase 4 (PAD4) Inhibitor
ACS Med. Chem. Lett.  20189, 1013–1018.
305. Boerth, J. A.; Maity, S.; Williams, S. K.; Mercado, B. Q.; Ellman, J. A.
Selective and Synergistic Cobalt(III)-Catalysed Three-Component C–H Bond Addition to Dienes and Aldehydes
Nat. Catal.  20181, 673–679.
304. Hoang, G. L.; Li, Y.; Halskov, K. S.; Ellman, J. A
Synthesis of Azolo[1,3,5]triazines via Rhodium(III)-Catalyzed Annulation of N-Azolo Imines and Dioxazolones
J. Org. Chem.  201883, 9522–9529.
303. Potter, T.J.; Li, Y.; Ward, M. D.; Ellman, J. A.
Rh(III)-Catalyzed Synthesis of Isoquinolones and 2-Pyridones via Annulation of N-Methoxyamides and Nitroalkenes
Eur. J. Org. Chem.  20182018, 4381–4388 [International Adivsory Board 20th Anniversary Issue].
302. Walker, M. M.; Chen, S.; Houk, K.; Ellman, J. A.
Formation of Aminocyclopentadienes from Silyldihydropyridines: Ring Contractions Driven by Anion Stabilization
Angew. Chem. Int. Ed.  201857, 6605–6609.
301. Hoang, G. L.; Ellman, J. A.
Rhodium(III)-Catalyzed C–H Functionalization of C-Alkenyl Azoles with Sulfoxonium Ylides for the Synthesis of Bridgehead N-Fused [5,6]-bicyclic Heterocycles
Tetrahedron  201874, 3318–3324 [Herzon Tetrahedron Young Investigator Award Issue].
Sigma/Aldrich technology spotlight and commercial availability of ketosulfoxonium ylides
300. Halskov, K. M.; Witten, M. R.; Hoang, G. L.; Mercado, B. Q.; Ellman, J. A.
Rhodium(III)-Catalyzed Imidoyl C−H Activation for Annulations to Azolopyrimidines
Org. Lett.  201820, 2464–2467.
Research Highlight in Synfacts, Sigma/Aldrich technology spotlight and commercial availability of ketosulfoxonium ylides
299. Xu, J.; Hartley, B. J.; Kurup, P.; Phillips, A.; Topol, A.; Xu, M.; Ononenyi, C.; Foscue, E.; Ho, S. M.; Baguley, T. D.; Carty, N.; Barros, C. S.; Müller, U.; Gupta, S.; Gochman, P.; Rapoport, J.; Ellman, J. A.; et al.
Inhibition of STEP61 Ameliorates Deficits in Mouse and hiPSC-Based Schizophrenia Models
Mol. Psychiatry  201823, 271–281.
298. Tjin, C. C.; Otley, K. D.; Baguley, T. D.; Kurup, P.; Xu, J.; Nairn, A. C.; Lombroso, P. J.; Ellman, J. A.
Glutathione-Responsive Selenosulfide Prodrugs as a Platform Strategy for Potent and Selective Mechanism-Based Inhibition of Protein Tyrosine Phosphatases
ACS Cent. Sci.  20173, 1322–1328.
297. Tran, G.; Confair, D.; Hesp, K. D.; Mascitti, V.; Ellman, J. A.
C2-Selective Branched Alkylation of Benzimidazoles by Rhodium(I)-Catalyzed C–H Activation
J. Org. Chem.  201782, 9243–9252.
296. Witten, M. R.; Wissler, L.; Snow, M.; Geschwindner, S.; Read, J. A.; Brandon, N. J.; Nairn, A. C.; Lombroso, P. J.; Käck, H.; Ellman, J. A.
X-ray Characterization and Structure-Based Optimization of Striatal-Enriched Protein Tyrosine Phosphatase Inhibitors
J. Med. Chem.  201760, 9299–9319.
295. Boerth, J. A.; Ellman, J. A.
A Convergent Synthesis of Functionalized Alkenyl Halides via Co(III)-Catalyzed Three-Component C-H Bond Addition
Angew. Chem. Int. Ed.  201756, 9976–9980 [Very Important Paper].
294. Halskov, K.; Roth, H.; Ellman, J. A.
Synthesis of [5,6]-Bicyclic Heterocycles with a Ring-Junction Nitrogen via Rh(III)-Catalyzed C-H Functionalization of Alkenyl Azoles
Angew. Chem. Int. Ed.  201756, 9183–9187.
293. Potter, T. J.; Ellman, J. A.
Total Synthesis of (+)-Pancratistatin by the Rh(III)-Catalyzed Addition of a Densely Functionalized Benzamide to a Sugar-Derived Nitroalkene
Org. Lett.  201719, 2985–2988.
292. Tran, G.; Hesp, K. D.; Mascitti, V.; Ellman, J. A.
Base-Controlled Completely Selective Linear or Branched Rhodium(I)-Catalyzed C−H ortho-Alkylation of Azines without Preactivation
Angew. Chem. Int. Ed.  201756, 5899–5903.
291. Hummel, J. R.; Boerth, J. A.; Ellman, J. A.
Transition-Metal-Catalyzed C–H Bond Addition to Carbonyls, Imines, and Related Polarized π Bonds
Chem. Rev.  2017117, 9163–9227.

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