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349. |
Goodner, R. M.; Brandes, D. S.; Morais, G. N.; Tao, Q.; Tassone, J. P.; Mercado, B. Q.; Chen, S.; Ellman, J. A.
C–H Activation and Sequential Addition to Dienes and Imines: Synthesis of Amines with β-Quaternary Centers and Mechanistic Studies on the Complex Interplay Between the Catalyst and Three Reactants
ACS Catal. 2024, 14, 18124–18133.
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348. |
Yeo, J.; Tassone, J. P.; Ellman, J. A.
Synthesis of α-Quaternary Amides via Cp*Co(III)-Catalyzed Sequential C–H Bond Addition to 1,3-Dienes and Isocyanates
Org. Lett. 2024, 26, 9769–9774.
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347. |
Molas, J. C.; Poag, E. M.; Ellman, J. A.
Synthesis of Monodehydro-Diketopiperazines Enabled by Cp*Rh(III)-Catalyzed Amine-Directed N–H Functionalization
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346. |
Moon, M. H.; Vock, I. W.; Streit, A. D.; Connor, L. J.; Senkina, J.; Ellman, J. A.; Simon, M. D.
Disulfide Tethering to Map Small Molecule Binding Sites Transcriptome-wide
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345. |
Champlin, A. T.; Kwon, N. Y.; Ellman, J. A.
Enantioselective S-Alkylation of Sulfenamides by Phase-Transfer Catalysis
Angew. Chem. Int. Ed. 2024, 63, e202408820.
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344. |
Patel, S.; Greenwood, N. S.; Mercado, B. Q.; Ellman, J. A.
Rh(II)-Catalyzed Enantioselective S-Alkylation of Sulfenamides with Acceptor–Acceptor Diazo Compounds Enables the Synthesis of Sulfoximines Displaying Diverse Functionality
Org. Lett. 2024, 26, 6295–6300.
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343. |
Chu, D.; Zoll, A. J.; Ellman, J. A.
Copper-Catalyzed Three-Component Synthesis of Highly Substituted Morpholines
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342. |
Greenwood, N. S.; Cerny, N. P.; Deziel, A. P.; Ellman, J. A.
Synthesis of N-Acylsulfenamides from (Hetero)Aryl Iodides and Boronic Acids by One-Pot Sulfur-Arylation and Dealkylation
Angew. Chem. Int. Ed. 2024, 63, e202315701.
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341. |
Vargas-Rivera, M. A.; Liu, A. S.; Ellman, J. A.
Visible-Light-Mediated, Diastereoselective Epimerization of Exocyclic Amines
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340. |
Greenwood, N. S.; Ellman, J. A.
Sulfur-Arylation of Sulfenamides via Ullmann-Type Coupling with (Hetero)aryl Iodides
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339. |
Champlin, A. T.; Ellman, J. A.
Preparation of Sulfilimines by Sulfur-Alkylation of N-Acyl Sulfenamides with Alkyl Halides
J. Org. Chem. 2023, 88, 7607–7614.
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338. |
Chu, D.; Ellman, J. A.
Stereospecific Synthesis of Unprotected, α,β-Disubstituted Tryptamines and Phenethylamines from 1,2-Disubstituted Alkenes via a One-Pot Reaction Sequence
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337. |
Greenwood, N. S.; Ellman, J. A.
Sulfur-Arylation of Sulfenamides via Chan–Lam Coupling with Boronic Acids: Access to High Oxidation State Sulfur Pharmacophores
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336. |
Liu, J. T.; Brandes, D. S.; Greenwood, N. S.; Ellman, J. A.
Synthesis of N-Acylsulfenamides from Amides and N-Thiosuccinimides
Synthesis 2023, 55, 2353–2360 [Special Issue dedicated to Prof. David A. Evans].
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335. |
Zoll, A. J.; Molas, J. C.; Mercado, B. Q.; Ellman, J. A.
Imine Directed Cp*Rh(III)-Catalyzed N–H Functionalization and Annulation with Amino Amides, Aldehydes, and Diazo Compounds
Angew. Chem. Int. Ed. 2023, 62, e202210822.
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334. |
Tassone, J. P.; Yeo, J. Ellman, J. A.
Three-component carboformylation: α-quaternary aldehyde synthesis via Co(III)-catalysed sequential C–H bond addition to dienes and acetic formic anhydride
Chem. Sci. 2022, 13, 14320–14326.
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333. |
Shen, Z.; Vargas-Rivera, M.; Rigby, E. L.; Chen, S.; Ellman, J. A.
Visible Light-Mediated, Highly Stereoselective Epimerization of Morpholines and Piperazines to the More Stable Isomers
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332. |
Kaplan, A.; Confair, D. N.; Kim, K.; Barros Álvarez, X.; Rodriguiz, R. M.; Yang, Y.; Kweon, O. S.; Che, T.; McCorvy, J.; Kamber, D. N.; Phelan, J. P. Martins, L. C.;...Wetsel, W. C.; Irwin, J. J.; Skiniotis, G.; Shoichet, B. K.; Roth, B. L.; Ellman, J. A.
Bespoke library docking for 5-HT2A receptor agonists with antidepressant activity
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331. |
Greenwood, N. S.; Champlin, A. T.; Ellman, J. A.
Catalytic Enantioselective Sulfur Alkylation of Sulfenamides for the Asymmetric Synthesis of Sulfoximines
J. Am. Chem. Soc. 2022, 144, 17808–17814.
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330. |
Gannam, Z. T. K.; Jamali, H.; Kweon, O. S.; Herrington, J.; Papini, C.; Gentzel, E.; Lolis, E.; Bennett, A. M.; Ellman, J. A.; Anderson, K. S.
Defining the Structure-Activity Relationship for a Novel Class of Allosteric MKP5 Inhibitors
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329. |
Brandes, D. S.; Ellman, J. A.
C–H bond activation and sequential addition to two different coupling partners: a versatile approach to molecular complexity
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328. |
Kazerouni, A. M.; Brandes, D. S.; Davies, C. C.; Cotter, L. F.; Mayer, J. M.; Chen, S.; Ellman, J. A.
Visible Light-Mediated, Highly Diastereoselective Epimerization of Lactams from the Most Accessible to the More Stable Stereoisomer
ACS Catal. 2022, 12, 7798–7803.
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327. |
Xu, C.; Tassone, J. P.; Mercado, B. Q.; Ellman, J. A.
Stereoselective Synthesis of Allenyl Alcohols by Cobalt(III)-Catalyzed Sequential C−H Bond Addition to 1,3-Enynes and Aldehydes
Angew. Chem. Int. Ed. 2022, 61, e202202364 [Hot Paper].
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326. |
Chu, D.; Ellman, J. A.
Three-Component Friedel–Crafts Transformations: Synthesis of Alkyl and Alkenyl Trifluoromethyl Sulfides and Alkenyl Iodides
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325. |
Brandes, D. S.; Muma, A. D.; Ellman, J. A.
Synthesis of α-Branched Amines by Three- and Four-Component C–H Functionalization Employing a Readily Diversifiable Hydrazone Directing Group
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Chen, S.; Chandra Tjin, C.; Gao, X.; Xue, Y.; Jiao, H.; Zhang, R.; Wu, M.; He, Z.; Ellman, J. A.; Ha, Y.
Pharmacological inhibition of PI5P4Kα/β disrupts cell energy metabolism and selectively kills p53-null tumor cells
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Brandes, D. S.; Sirvent, A.; Mercado, B. Q.; Ellman, J. A.
Three-Component 1,2-Carboamidation of Bridged Bicyclic Alkenes via RhIII-Catalyzed Addition of C–H Bonds and Amidating Reagents
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322. |
Dongbang, S.; Confair, D. N.; Ellman, J. A.
Rhodium-Catalyzed C–H Alkenylation/Electrocyclization Cascade Provides Dihydropyridines That Serve as Versatile Intermediates to Diverse Nitrogen Heterocycles
Acc. Chem. Res. 2021, 54, 1766-1778.
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Shen, Z.; Walker, M. M.; Chen, S.; Parada, G. A.; Chu, D. M.; Dongbang, S.; Mayer, J. M.; Houk, K. N.; Ellman, J. A.
General Light-Mediated, Highly Diastereoselective Piperidine Epimerization: From Most Accessible to Most Stable Stereoisomer
J. Am. Chem. Soc. 2021, 143, 126–131.
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320. |
Dongbang, S.; Ellman, Jonathan A.
Synthesis of Nitrile Bearing Acyclic Quaternary Centers via Co(III)‐Catalyzed Sequential C–H Bond Addition to Dienes and N‐Cyanosuccinimide
Angew. Chem. Int. Ed. 2021, 60, 2135-2139.
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