Publications
| 42. |
Boojamra, C. G.; Burow, K. M.; Thompson, L. A.; Ellman, J. A. The Solid-Phase Synthesis of 1,4-Benzodiazepine-2,5-diones. Library Preparation and Demonstration of Synthesis Generality J. Org. Chem. 1997, 62, 1240-1257. |
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| 41. |
Plunkett, M. J.; Ellman, J. A. Combinatorial Chemistry and New Drugs Sci. Am. 1997, 276, 68-73. |
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| 40. |
Plunkett, M. J.; Ellman, J. A. “Combinatorial Chemistry” in McGraw-Hill Yearbook of Science & Technology, Parker, S. P., Ed.; McGraw-Hill Book Co.: New York, New York, 1997, , 95-99. |
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| 39. |
Bunin, B. A.; Plunkett, M. J.; Bray, A. M.; Ellman, J. A. The Synthesis of a 1680 Compound 1,4-Benzodiazepine Library New J. Chem. 1997, 21, 125. |
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| 38. |
Choong, I. C.; Ellman, J. A. Solid-Phase Synthesis: Application of Combinatorial Libraries in Annu. Rep. Med. Chem. 1996, 31, 309-318. |
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| 37. |
Stevens, S. Y.; Bunin, B. A.; Plunkett, M. J.; Swanson, P. C.; Ellman, J. A.; Glick, G. D. Non-Nucleic Acid Inhibitors of Protein-DNA Interactions Identified through Combinatorial Chemistry J. Am. Chem. Soc. 1996, 118, 10650-10651. |
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| 36. |
Virgilio, A. A.; Schürer, S.; Ellman, J. A Expedient Synthesis of beta-Turn Mimetics Incorporating the i + 1, i + 2, and i + 3 Sidechains Tetrahedron Lett. 1996, 37, 6961-6964. |
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| 35. |
Backes, B. J.; Virgilio, A. A.; Ellman, J. A Activation Method to Prepare a Highly Reactive Acylsulfonamide “Safety-Catch” Linker for Solid-Phase Synthesis J. Am. Chem. Soc. 1996, 118, 3055-3057. |
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| 34. |
Koh, J. S.; Ellman, J. A Palladium-Mediated Three-Component Coupling Strategy for the Solid-Phase Synthesis of Tropane Derivatives J. Org. Chem. 1996, 61, 4494-4495. |
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| 33. |
Virgilio, A. A.; Ellman, J. A. “Conformationally Restricted Peptide and Peptidomimetic Libraries” in Combinatorial Chemistry and Molecular Diversity in Drug Discovery; Gordon, E. M. and Kerwin, J. F. Ed.; John Wiley & Sons, Inc.: New York, New York, 1998, , 133-151. |
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| 32. |
Ellman, J. A The Solid-Phase Synthesis of Complex Small Molecules Chimia 1996, 50, 260-261. |
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| 31. |
Ellman, J. A Design, Synthesis, and Evaluation of Small-Molecule Libraries Acc. Chem. Res. 1996, 29, 132-143. |
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| 30. |
Thompson, L. A.; Ellman, J. A. Synthesis and Applications of Small Molecule Libraries Chem. Rev. 1996, 96, 555-600. |
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| 29. |
Bunin, B. A.; Plunkett, M. J.; Ellman, J. A. Synthesis and Evaluation of 1,4-Benzodiazepine Libraries Methods Enzymol. 1996, 267, 448-467. |
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| 28. |
Liu, G.; Ellman, J. A. A General Solid-Phase Synthesis Strategy for the Preparation of 2-Pyrrolidinemethanol Ligands J. Org. Chem. 1995, 60, 7712–7713. |
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| 27. |
Plunkett, M. J.; Ellman, J. A Silicon-Based Linkage Strategy for Traceless Solid-Phase Synthesis J. Org. Chem. 1995, 60, 6006-6007. |
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| 26. |
Boojamra, C G.; Burow, K. J.; Ellman, J. A A General and Straightforward Method for the Solid-Phase Synthesis of 1,4-Benzodiazepine-2,5-diones J. Org. Chem. 1995, 60, 5742-5743. |
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| 25. |
Ellman, J. A. “Synthesis and Evaluation of 1,4-Benzodiazepine Libraries” in Combinatorial Peptide and Nonpeptide Libraries; Jung, G. Ed.; VCH Verlagsgesellschaft mbH: Weinham, Germany 1996, , 405-424. |
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| 24. |
Ellman, J. A Combinatorial Organic Libraries CHEMTRACTS: Org. Chem 1995, 8, 1-4. |
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| 23. |
Kick, E. K.; Ellman, J. A Expedient Method for the Solid-Phase Synthesis of Aspartic Acid Protease Inhibitors Directed toward the Generation of Libraries J. Med. Chem. 1995, 38, 1427-1430. |
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| 22. |
Plunkett, M. J.; Ellman, J. A Stille Coupling in the Solid-Phase Synthesis of Structurally Diverse 1,4-Benzodiazepine Derivatives J. Am. Chem. Soc. 1995, 117, 3306-3307. |
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| 21. |
Thompson, L. A.; Ellman, J. A Straightforward and General Method for Coupling Alcohols to Solid-Supports Tetrahedron Lett. 1994, 35, 9333-9336. |
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| 20. |
Virgilio, A. A.; Ellman, J. A Simultaneous Solid-Phase Synthesis of beta-Turn Mimetics Incorporating Side-Chain Functionality J. Am. Chem. Soc. 1994, 116, 11580-11581. |
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| 19. |
Backes, B. J.; Ellman, J. A Carbon-Carbon Bond Forming Methods on Solid Support. Utilization of Kenner’s “Safety-Catch” Linker J. Am. Chem. Soc. 1994, 116, 11171-11172. |
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| 18. |
Bunin, B. A.; Ellman, J. A. Increasing the Diversity of a 1,4-Benzodiazepine Library through Side-Chain Functionalization Polym. Prepr. 1994, 35, 983. |
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| 17. |
Bunin, B. A.; Plunkett, M. J.; Ellman, J. A The Combinatorial Synthesis, and Chemical and Biological Evaluation of a 1,4-Benzodiazepine Library Proc. Natl. Acad. Sci USA 1994, 91, 4708-4712. |
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| 16. |
Bunin, B. A.; Ellman, J. A. A General and Expedient Method for the Solid-Phase Synthesis of 1,4-Benzodiazepine Derivatives J. Am. Chem. Soc. 1992, 114, 10997-10998. |
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| 14. |
Cook, S. N.; Jack, W. E.; Xiong, X.; Danley, L. E.; Ellman, J. A.; Schultz, P. G.; Noren, C. J. Photochemically-Initiated Protein Splicing Angew. Chem., Int. Ed. Engl. 1995, 34, 1629-1630. |
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| 13. |
Mendel, D.; Ellman, J. A.; Schultz, P. G. Protein Biosynthesis with Conformationally Restricted Amino Acids J. Am. Chem. Soc. 1993, 115, 4359-4360. |
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| 12. |
Ellman, J. A.; Volkman, B. F.; Mendel, D.; Schultz, P. G.; Wemmer, D. E Site-Specific Isotopic Labeling of Proteins for NMR Studies J. Am. Chem. Soc. 1992, 114, 7959-7961. |