Publications
| 50. |
Woolard, F. X.; Paetsch, J.; Ellman, J. A. A Silicon Linker for the Direct Loading of Aromatic Compounds onto Solid Supports. Traceless Synthesis of Pyridyl-Based Tricyclics J. Org. Chem. 1997, 62, 6102-6103. |
|
| 49. |
Liu, G.; Cogan, D. A.; Ellman, J. A Catalytic Asymmetric Synthesis of tert-Butanesulfinamide. Application to the Asymmetric Synthesis of Amines J. Am. Chem. Soc. 1997, 119, 9913-9914. |
|
| 48. |
Backes, B. A.; Ellman, J. A. Solid Support Linker Strategies Curr. Opin. Chem. Biol. 1997, 1, 86-94. |
|
| 47. |
Kick, E. K.; Roe, D. C.; Skillman, A. G.; Liu, G.; Ewing, T. J. A.; Sun, Y.; Kuntz, I. D.; Ellman, J. A. Structure-Based Design and Combinatorial Chemistry Yield Low Nanomolar Inhibitors of Cathepsin D Chem. Biol. 1997, 4, 297-309. |
|
| 46. |
Virgilio, A. A.; Bray, A. A.; Zhang, W.; Ellman, J. A. Synthesis and Evaluation of a Library of Peptidomimetics Based upon the beta-Turn Tetrahedron 1997, 53, 6635-6644. |
|
| 45. |
Plunkett, M. J.; Ellman, J. A. Germanium and Silicon Linking Strategies for Traceless Solid-Phase Synthesis J. Org. Chem. 1997, 62, 2885-2893. |
|
| 44. |
Ellman, J. Stoddard, B.; Wells, J. Combinatorial Thinking in Chemistry and Biology Proc. Natl. Acad. Sci., USA 1997, 94, 2779-2782. |
|
| 43. |
Evans, D. A.; Barrow, J. C.; Watson, P. S.; Ratz, A. M.; Dinsmore, C. J.; Evrard, D. A.; DeVries, K.; Ellman, J. A.; Rychnovsky, S. D.; Lacour, J Synthesis and Conformational Properties of the M(4-6)(5-7) Bicyclic Tetrapeptide Common to the Vancomycin Antibiotics J. Am. Chem. Soc. 1997, 119, 3419-3420. |
|
| 42. |
Boojamra, C. G.; Burow, K. M.; Thompson, L. A.; Ellman, J. A. The Solid-Phase Synthesis of 1,4-Benzodiazepine-2,5-diones. Library Preparation and Demonstration of Synthesis Generality J. Org. Chem. 1997, 62, 1240-1257. |
|
| 41. |
Plunkett, M. J.; Ellman, J. A. Combinatorial Chemistry and New Drugs Sci. Am. 1997, 276, 68-73. |
|
| 40. |
Plunkett, M. J.; Ellman, J. A. “Combinatorial Chemistry” in McGraw-Hill Yearbook of Science & Technology, Parker, S. P., Ed.; McGraw-Hill Book Co.: New York, New York, 1997, , 95-99. |
|
| 39. |
Bunin, B. A.; Plunkett, M. J.; Bray, A. M.; Ellman, J. A. The Synthesis of a 1680 Compound 1,4-Benzodiazepine Library New J. Chem. 1997, 21, 125. |
|
| 38. |
Choong, I. C.; Ellman, J. A. Solid-Phase Synthesis: Application of Combinatorial Libraries in Annu. Rep. Med. Chem. 1996, 31, 309-318. |
|
| 37. |
Stevens, S. Y.; Bunin, B. A.; Plunkett, M. J.; Swanson, P. C.; Ellman, J. A.; Glick, G. D. Non-Nucleic Acid Inhibitors of Protein-DNA Interactions Identified through Combinatorial Chemistry J. Am. Chem. Soc. 1996, 118, 10650-10651. |
|
| 36. |
Virgilio, A. A.; Schürer, S.; Ellman, J. A Expedient Synthesis of beta-Turn Mimetics Incorporating the i + 1, i + 2, and i + 3 Sidechains Tetrahedron Lett. 1996, 37, 6961-6964. |
|
| 35. |
Backes, B. J.; Virgilio, A. A.; Ellman, J. A Activation Method to Prepare a Highly Reactive Acylsulfonamide “Safety-Catch” Linker for Solid-Phase Synthesis J. Am. Chem. Soc. 1996, 118, 3055-3057. |
|
| 34. |
Koh, J. S.; Ellman, J. A Palladium-Mediated Three-Component Coupling Strategy for the Solid-Phase Synthesis of Tropane Derivatives J. Org. Chem. 1996, 61, 4494-4495. |
|
| 33. |
Virgilio, A. A.; Ellman, J. A. “Conformationally Restricted Peptide and Peptidomimetic Libraries” in Combinatorial Chemistry and Molecular Diversity in Drug Discovery; Gordon, E. M. and Kerwin, J. F. Ed.; John Wiley & Sons, Inc.: New York, New York, 1998, , 133-151. |
|
| 32. |
Ellman, J. A The Solid-Phase Synthesis of Complex Small Molecules Chimia 1996, 50, 260-261. |
|
| 31. |
Ellman, J. A Design, Synthesis, and Evaluation of Small-Molecule Libraries Acc. Chem. Res. 1996, 29, 132-143. |
|
| 30. |
Thompson, L. A.; Ellman, J. A. Synthesis and Applications of Small Molecule Libraries Chem. Rev. 1996, 96, 555-600. |
|
| 29. |
Bunin, B. A.; Plunkett, M. J.; Ellman, J. A. Synthesis and Evaluation of 1,4-Benzodiazepine Libraries Methods Enzymol. 1996, 267, 448-467. |
|
| 28. |
Liu, G.; Ellman, J. A. A General Solid-Phase Synthesis Strategy for the Preparation of 2-Pyrrolidinemethanol Ligands J. Org. Chem. 1995, 60, 7712–7713. |
|
| 27. |
Plunkett, M. J.; Ellman, J. A Silicon-Based Linkage Strategy for Traceless Solid-Phase Synthesis J. Org. Chem. 1995, 60, 6006-6007. |
|
| 26. |
Boojamra, C G.; Burow, K. J.; Ellman, J. A A General and Straightforward Method for the Solid-Phase Synthesis of 1,4-Benzodiazepine-2,5-diones J. Org. Chem. 1995, 60, 5742-5743. |
|
| 25. |
Ellman, J. A. “Synthesis and Evaluation of 1,4-Benzodiazepine Libraries” in Combinatorial Peptide and Nonpeptide Libraries; Jung, G. Ed.; VCH Verlagsgesellschaft mbH: Weinham, Germany 1996, , 405-424. |
|
| 24. |
Ellman, J. A Combinatorial Organic Libraries CHEMTRACTS: Org. Chem 1995, 8, 1-4. |
|
| 23. |
Kick, E. K.; Ellman, J. A Expedient Method for the Solid-Phase Synthesis of Aspartic Acid Protease Inhibitors Directed toward the Generation of Libraries J. Med. Chem. 1995, 38, 1427-1430. |
|
| 22. |
Plunkett, M. J.; Ellman, J. A Stille Coupling in the Solid-Phase Synthesis of Structurally Diverse 1,4-Benzodiazepine Derivatives J. Am. Chem. Soc. 1995, 117, 3306-3307. |
|
| 21. |
Thompson, L. A.; Ellman, J. A Straightforward and General Method for Coupling Alcohols to Solid-Supports Tetrahedron Lett. 1994, 35, 9333-9336. |