Publications

297. Tran, G.; Confair, D.; Hesp, K. D.; Mascitti, V.; Ellman, J. A.
C2-Selective Branched Alkylation of Benzimidazoles by Rhodium(I)-Catalyzed C–H Activation
J. Org. Chem.  201782, 9243–9252.  
296. Boerth, J. A.; Ellman, J. A.
A Convergent Synthesis of Functionalized Alkenyl Halides via Co(III)-Catalyzed Three-Component C-H Bond Addition
Angew. Chem. Int. Ed.  201756, 9976–9980.  
295. Hummel, J. R.; Ellman, J. A.
Convergent Synthesis of α-Branched Amines by Transition-Metal-Catalyzed C−H Bond Additions to Imines
Isr. J. Chem.  201757, Early View.  
294. Halskov, K.; Roth, H.; Ellman, J. A.
Synthesis of [5,6]-Bicyclic Heterocycles with a Ring-Junction Nitrogen via Rh(III)-Catalyzed C-H Functionalization of Alkenyl Azoles
Angew. Chem. Int. Ed.  201756, 9183–9187.  
293. Potter, T. J.; Ellman, J. A.
Total Synthesis of (+)-Pancratistatin by the Rh(III)-Catalyzed Addition of a Densely Functionalized Benzamide to a Sugar-Derived Nitroalkene
Org. Lett.  201719, 2985–2988.  
292. Tran, G.; Hesp, K. D.; Mascitti, V.; Ellman, J. A.
Base-Controlled Completely Selective Linear or Branched Rhodium(I)-Catalyzed C−H ortho-Alkylation of Azines without Preactivation
Angew. Chem. Int. Ed.  201756, 5899–5903.  
291. Hummel, J. R.; Boerth, J. A.; Ellman, J. A.
Transition-Metal-Catalyzed C–H Bond Addition to Carbonyls, Imines, and Related Polarized π Bonds
Chem. Rev.  2017117, 9163–9227.  
290. Potter, T. J.; Kamber, D. N.; Mercado, B. Q.; Ellman, J. A.
Rh(III)-Catalyzed Aryl and Alkenyl C–H Bond Addition to Diverse Nitroalkenes
ACS Catal.  20177, 150–153.  
289. Xu, J.; Hartley, B. J.; Kurup, P.; Phillips, A.; Topol, A.; Xu, M.; Ononenyi, C.; Foscue, E.; Ho, S. M.; Baguley, T. D.; Carty, N.; Barros, C. S.; Müller, U.; Gupta, S.; Gochman, P.; Rapoport, J.; Ellman, J. A.; et al.
Inhibition of STEP61 Ameliorates Deficits in Mouse and hiPSC-Based Schizophrenia Models
Mol. Psychiatry  2017Epub ahead of print, .  
288. Wangweerawong, A.; Kolmar. S.; Ellman, J. A.
Preparation of (S)-Nonafluorobutanesulfinamide
Org. Synth.  201693, 319-330.  
287. Chen, S.; Bacauanu, V.; Knecht, T.; Mercado, B. Q.; Bergman, R. G.; Ellman, J. A.
New Regio- and Stereoselective Cascades via Unstabilized Azomethine Ylide Cycloadditions for the Synthesis of Highly Substituted Tropane and Indolizidine Frameworks
J. Am. Chem. Soc.  2016138, 12664–12670.  
286. Potter, T. J.; Ellman, J. A.
Rh(III)-Catalyzed C–H Bond Addition/Amine-Mediated Cyclization of Bis-Michael Acceptors
Org. Lett.  201618, 3838–3841.  
285. Jamali, H.; Khan, H. A.; Tjin, C. C.; Ellman, J. A.
Cellular Activity of New Small Molecule Protein Arginine Deiminase 3 (PAD3) Inhibitors
ACS Med. Chem. Lett.  20167, 847–851.  
284. Weinstein, A. B.; Ellman, J. A.
Convergent Synthesis of Diverse Nitrogen Heterocycles via Rh(III)-Catalyzed C–H Conjugate Addition/Cyclization Reactions
Org. Lett.  201618, 3294-3297.  
283. Boerth, J. A.; Hummel, J. R.; Ellman, J. A.
Highly Stereoselective Cobalt(III)-Catalyzed Three-Component C−H Bond Addition Cascade
Angew. Chem. Int. Ed.  201655, 12650-12654.  
282. Phelan, J. P.; Ellman, J. A.
Conjugate Addition–Enantioselective Protonation Reactions
Beilstein J. Org. Chem.  201612, 1203–1228.  
281. Mesganaw, T.; Elman, J. A.
4-(Diethylphosphino)-N,N-dimethylaniline
e-EROS Encyclopedia of Reagents for Organic Synthesis  2016, .  
280. Phelan, J. P.; Ellman, J. A.
Catalytic Enantioselective Addition of Pyrazol-5-ones to Trisubstituted Nitroalkenes with an N-Sulfinylurea Organocatalyst
Adv. Synth. Catal.  2016358, 1713–1718.  
279. Wangweerawong, A.; Hummel, J. R.; Bergman, R. G.; Ellman, J. A.
Preparation of Enantiomerically Pure Perfluorobutanesulfinamide and Its Application to the Asymmetric Synthesis of α-Amino Acids
J. Org. Chem.  201681, 1547–1557.  
278. Boerth, J. A.; Ellman, J. A.
Rh(III)-Catalyzed Diastereoselective C–H Bond Addition/Cyclization Cascade of Enone Tethered Aldehydes
Chem. Sci.  20167, 1474-1479.  
277. Xu, J.; Kurup, P.; Baguley, T.; Foscue, E.; Ellman J. A.; Nairn, A. C.; Lombroso, P. J.
Inhibition of the Tyrosine Phosphatase STEP61 Restores BDNF Expression and Reverses Motor and Cognitive Deficits in Phencyclidine-Treated Mice
Cell. Mol. Life Sci.  201673, 1503-1514.  
276. Azkona, G.; Saavedra, A.; Aira, Z.; Aluja, D.; Xifró, X.; Baguley, T.; Alberch, J.; Ellman J. A.; Lombroso, P. J.; Azkue, J. J.; Pérez-Navarro, E.
Striatal-Enriched Protein Tyrosine Phosphatase Modulates Nociception: Evidence from Genetic Deletion and Pharmacological Inhibition
Pain  2016157, 377-86.  
275. Xu, J.; Kurup, P. K.; Azkona, G. M.; Baguley, T. D.; Saavedra, A. C.; Nairn, A. C.; Ellman, J. A.; Perez-Navarro, E.; Lombroso, P. A.
Down-Regulation of BDNF in Cell and Animal Models Increases Striatal-Enriched Protein Tyrosine Phosphatase STEP61 Levels
J. Neurochem.  2016136, 285–294.  
274. Phillips, E. M.; Mesganaw, T.; Patel, A. Duttwyler, S.; Mercado, B. Q.; Houk, K. N.; Ellman, J. A.
Synthesis of ent-Ketorfanol via a C–H Alkenylation/ Torquoselective 6π-Electrocyclization Cascade
Angew. Chem. Int. Ed.  201554, 12044–12048.  
273. Neitz, R. J.; Bryant, C.; Chen, S.; Gut, J.; Caselli, E. H.; Ponce, S.; Chowdhury, S.; Xu, H.; Arkin, M. R.; Ellman, J. A.; Renslo, A. R.
Tetrafluorophenoxymethyl Ketone Cruzain Inhibitors with Improved Pharmacokinetic Properties as Therapeutic Leads for Chagas’ Disease
Bioorg. Med. Chem. Lett.   201525, 4834–4837.  
272. Chen, S.; Mercado, B. Q.; Bergman, R. G.; Ellman, J. A.
Regio- and Diastereoselective Synthesis of Highly Substituted, Oxygenated Piperidines from Tetrahydropyridines
J. Org. Chem.  201580, 6660–6668.  
271. Chen, S.; Bergman, R. G.; Ellman, J. A.
Facile Rh(III)-Catalyzed Synthesis of Fluorinated Pyridines
Org. Lett.  201517, 2567–2569.  
270. Hummel, J. R.; Ellman, J. A.
Cobalt(III)-Catalyzed C–H Bond Amidation with Isocyanates
Org. Lett.  201517, 2400–2403.  
269. Oresic Bender, K.; Ofori, L.; van der Linden, W. A.; Mock, E. D.; Datta, G.; Chowdhury, S.; Li, H.; Segal, E.; Lopez, M. S.; Ellman, J. A.; Figdor, C. G.; Bogyo, M.; Verdoes, M.
Design of a Highly Selective Quenched Activity-Based Probe and Its Application in Dual Color Imaging Studies of Cathepsin S Activity Localization
J. Am. Chem. Soc.  2015137, 4771–4777.  
268. Jamali, H.; Khan, H. A.; Stringer, J. A.; Chowdhury, S. Ellman, J. A.
Identification of Multiple Structurally-Distinct, Nonpeptidic Small Molecule Inhibitors of Protein Arginine Deiminase 3 Using a Substrate-Based Fragment Method
J. Am. Chem. Soc.   2015137, 3616–3621.  

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